SCHEMBL5770027

SCHEMBL5770027

CCOC(=O)Oc1[nH]c2cccc(F)c2c1C#N

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.38
HTT P42858 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
NLRP3 Q96P20 1/20 0.36
KDM4E B2RXH2 4/20 0.36
TSHR P16473 3/20 0.36
HSD17B10 Q99714 3/20 0.36
GLA P06280 3/20 0.36
GAA P10253 3/20 0.36
HPGD P15428 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
ALOX15 P16050 2/20 0.36
ATM Q13315 1/20 0.36
KMT2A Q03164 2/20 0.35
CXCR2 P25025 1/20 0.35
MEN1 O00255 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5766840 0.88 KDM4E (0.37) ALDH1A1HTTNPSR1RXFP1NLRP3
SCHEMBL9573823 0.73 CDK1 (0.39) ALDH1A1NLRP3KDM4EHSD17B10GAA
SCHEMBL5767967 0.72 ALDH1A1 (0.44) ALDH1A1RXFP1KDM4EHSD17B10GAA
SCHEMBL4705953 0.70 DAO (0.47) ALDH1A1KDM4EKMT2AMEN1MAPT
SCHEMBL9573863 0.70 CDK1 (0.39) ALDH1A1KDM4EHSD17B10GAAHPGD
SCHEMBL9232719 0.70 KDM4E (0.41) ALDH1A1NLRP3KDM4EHSD17B10GAA
SCHEMBL9573812 0.68 GAA (0.35) ALDH1A1GAAHPGDCYP1A2CYP2C19
SCHEMBL9573874 0.68 KDM4E (0.40) ALDH1A1KDM4EHSD17B10ALOX15KMT2A
SCHEMBL27215072 0.68 NLRP3 (0.46) ALDH1A1NLRP3KDM4ETSHRHSD17B10
SCHEMBL9937270 0.68 NPC1 (0.52) ALDH1A1HTTNPSR1KDM4ETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1625129-A1 HETEROCYCLYL-SUBSTITUTED DIHYDROQUINAZOLINES AND USE THEREOF AS AN ANTIVIRAL AGENT Bayer HealthCare AG (DE) 2006-02-15 EP disclosed
WO-2004099212-A1 HETEROCYCLYL-SUBSTITUTED DIHYDROQUINAZOLINES AND USE THEREOF AS AN ANTIVIRAL AGENT BAYER HEALTHCARE AG (DE) 2004-11-18 WO disclosed