SCHEMBL5773512

SCHEMBL5773512

CC(C)=C(F)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 4/20 0.44
CES2 O00748 3/20 0.44
TSHR P16473 3/20 0.39
ALDH1A1 P00352 2/20 0.39
DAO P14920 1/20 0.39
NAPRT Q6XQN6 1/20 0.39
ESR1 P03372 1/20 0.38
MAPT P10636 2/20 0.37
PTPN1 P18031 1/20 0.37
GSK3B P49841 1/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
LMNA P02545 1/20 0.37
MAPK1 P28482 1/20 0.37
HTT P42858 1/20 0.37
F2 P00734 1/20 0.36
F10 P00742 1/20 0.36
F12 P00748 1/20 0.36
F7 P08709 1/20 0.36
F3 P13726 1/20 0.36
PKM P14618 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16453535 0.83 CES1 (0.44) CES1CES2TSHRALDH1A1DAO
SCHEMBL16933810 0.83 CES1 (0.44) CES1CES2TSHRALDH1A1DAO
SCHEMBL3929950 0.82 CES1 (0.47) CES1CES2TSHRALDH1A1DAO
SCHEMBL18985177 0.82 CES1 (0.47) CES1CES2TSHRALDH1A1DAO
SCHEMBL2234110 0.82 CES1 (0.47) CES1CES2TSHRALDH1A1DAO
SCHEMBL4647631 0.77
SCHEMBL285854 0.77 CES1 (0.43) CES1CES2TSHRALDH1A1DAO
SCHEMBL22745485 0.76 ALDH1A1 (0.46) CES1CES2ALDH1A1MAPTGSK3B
SCHEMBL17847697 0.75 CES1 (0.48) CES1CES2TSHRALDH1A1DAO
Fluoride SCHEMBL8219548 0.74 CES1 (0.41) CES1CES2TSHRALDH1A1DAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1736471-B1 3-(DIHYDRO(TETRAHYDRO)ISOQUINOLIN-1-YL)QUINOLINES MITSUI CHEMICALS AGRO INC (JP) 2014-01-08 EP disclosed
EP-1736471-A1 3-(DIHYDRO(TETRAHYDRO)ISOQUINOLIN-1-YL)QUINOLINES Sankyo Agro Company, Limited (JP) 2006-12-27 EP disclosed