SCHEMBL5776112

SCHEMBL5776112

COc1c(F)cccc1C(C)(C)CC(O)C(F)(F)F

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CETP P11597 2/20 0.33
CTSS P25774 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
KCNH2 Q12809 1/20 0.33
NR3C1 P04150 2/20 0.32
NR3C2 P08235 2/20 0.32
PGR P06401 1/20 0.32
AR P10275 1/20 0.31
KMT2A Q03164 1/20 0.31
MGLL Q99685 1/20 0.30
GPBAR1 Q8TDU6 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3532509 0.73 NR3C1 (0.46) NR3C1NR3C2PGR
SCHEMBL23886230 0.73 KMT2A (0.37) CTSSSLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL31697313 0.72 AR (0.44) CTSSSLC6A2SLC6A4ARKMT2A
SCHEMBL22208564 0.72 AR (0.44) CTSSSLC6A2SLC6A4ARKMT2A
SCHEMBL13310501 0.72 CA2 (0.41) SLC6A2SLC6A4SLC6A3KCNH2AR
SCHEMBL3532136 0.72 CYP2D6 (0.35) CTSSNR3C1NR3C2PGR
SCHEMBL3536311 0.71 KRAS (0.37) CTSSSLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL3657310 0.71 NR3C2 (0.53) NR3C1NR3C2PGR
SCHEMBL1634224 0.71 NR3C2 (0.44) NR3C1NR3C2PGR
SCHEMBL3532410 0.71 NR3C1 (0.42) NR3C1NR3C2PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1638945-A1 HETEROCYCLICALLY SUBSTITUTED PENTANOL DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF, AND USE THEREOF AS ANTI-INFLAMMATORY AGENTS Schering Aktiengesellschaft (DE) 2006-03-29 EP disclosed
WO-2005003098-A1 HETEROCYCLICALLY SUBSTITUTED PENTANOL DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF, AND USE THEREOF AS ANTI-INFLAMMATORY AGENTS SCHERING AKTIENGESELLSCHAFT (DE) 2005-01-13 WO disclosed