SCHEMBL5776486

SCHEMBL5776486

CC(C)c1csc(C=Cc2cccc(N)c2C(=O)[C@@H]2OC(C)(C)O[C@H]2C(=O)O)n1

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALB P02768 1/20 0.39
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
GRM1 Q13255 1/20 0.33
CSNK2A2 P19784 1/20 0.31
CSNK2B P67870 1/20 0.31
CSNK2A1 P68400 1/20 0.31
CSNK2A3 Q8NEV1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5778590 0.83 ALB (0.40) ALBCYP1A2CYP2D6CYP2C9GRM1
SCHEMBL5778983 0.82 ALB (0.39) ALBCYP1A2CYP2D6CYP2C9GRM1
SCHEMBL5777697 0.82 ALB (0.39) ALBCYP1A2CYP2D6CYP2C9GRM1
SCHEMBL5776470 0.77 ALB (0.57) ALBCYP1A2CYP2D6CYP2C9GRM1
SCHEMBL5777728 0.71 ALB (0.43) ALBCYP1A2CYP2D6CYP2C9GRM1
SCHEMBL5779055 0.68 ALB (0.40) ALBCYP1A2
SCHEMBL5779934 0.66 NPC1 (0.31)
SCHEMBL5777537 0.64 ALB (0.47) ALBCYP1A2CYP2D6CYP2C9GRM1
SCHEMBL5779807 0.64 ALB (0.61) ALB
SCHEMBL5774563 0.63 ALB (0.69) ALB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1652839-A2 Drug efflux pump inhibitor DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2006-05-03 EP disclosed
EP-1227084-B1 DRUG DISCHARGE PUMP INHIBITORS TRINE PHARMACEUTICALS INC (US) 2005-12-14 EP disclosed