SCHEMBL5777697

SCHEMBL5777697

CC(C)c1csc(C=Cc2cccc(N)c2C(=O)[C@@H]2CCCC[C@H]2C(=O)O)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALB P02768 1/20 0.39
ALDH1A1 P00352 4/20 0.35
USP2 O75604 1/20 0.34
KDM4E B2RXH2 3/20 0.32
RAB9A P51151 3/20 0.32
NPC1 O15118 2/20 0.32
NPSR1 Q6W5P4 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
POLB P06746 1/20 0.32
CASP6 P55212 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
GRM1 Q13255 1/20 0.31
TAAR1 Q96RJ0 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
TP53 P04637 1/20 0.31
ADRB1 P08588 1/20 0.31
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5778983 1.00 ALB (0.39) ALBALDH1A1USP2KDM4ERAB9A
SCHEMBL5778590 0.90 ALB (0.40) ALBKMT2ACYP1A2CYP2D6CYP2C9
SCHEMBL5776486 0.82 ALB (0.39) ALBCYP1A2CYP2D6CYP2C9GRM1
SCHEMBL5778978 0.75 ALB (0.58) ALBALDH1A1USP2KDM4ERAB9A
SCHEMBL5777169 0.75 ALB (0.58) ALBALDH1A1USP2KDM4ERAB9A
SCHEMBL5779055 0.69 ALB (0.40) ALBALDH1A1KDM4ERAB9AMEN1
SCHEMBL5778584 0.67 ALB (0.60) ALBALDH1A1KDM4EMEN1KMT2A
SCHEMBL5777537 0.64 ALB (0.47) ALBALDH1A1KDM4ERAB9ANPC1
SCHEMBL5774563 0.63 ALB (0.69) ALBALDH1A1KDM4ERAB9ANPC1
SCHEMBL14759148 0.62 ALB (0.36) ALBRAB9AMEN1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1652839-A2 Drug efflux pump inhibitor DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2006-05-03 EP disclosed
EP-1227084-B1 DRUG DISCHARGE PUMP INHIBITORS TRINE PHARMACEUTICALS INC (US) 2005-12-14 EP disclosed