SCHEMBL5776526

SCHEMBL5776526

COC(=O)c1cc(OCCNC(=O)OC(C)(C)C)cc(C(=O)Nc2cccc(C=Cc3nc(-c4ccccc4)cs3)c2)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SNCA P37840 1/20 0.39
SUCNR1 Q9BXA5 5/20 0.39
HDAC3 O15379 4/20 0.37
HDAC1 Q13547 3/20 0.37
HDAC2 Q92769 3/20 0.37
HDAC10 Q969S8 3/20 0.37
HDAC8 Q9BY41 2/20 0.37
MAPT P10636 3/20 0.37
KDM4E B2RXH2 2/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
TP53 P04637 1/20 0.37
ADRB1 P08588 1/20 0.37
CYP3A4 P08684 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
HPGD P15428 1/20 0.37
PTGS1 P23219 1/20 0.37
KMT2A Q03164 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5781021 0.94 NR1H4 (0.41) SNCASUCNR1HDAC3HDAC1HDAC2
SCHEMBL5779901 0.83 ALB (0.51) SNCASUCNR1MAPTKDM4EMEN1
SCHEMBL5778188 0.76 ALB (0.52) SNCAMAPTKDM4EMEN1ALDH1A1
SCHEMBL5775504 0.74 ALB (0.49) SNCAMAPTKDM4EMEN1ALDH1A1
SCHEMBL5776928 0.71 ALB (0.57) SNCAMAPTKDM4EMEN1ALDH1A1
SCHEMBL5779176 0.71 CA12 (0.54) MAPTALDH1A1RAB9ANPC1
SCHEMBL9514907 0.69 ALB (0.48) MAPTKDM4EMEN1ALDH1A1TP53
SCHEMBL9518092 0.69 MAPT (0.50) MAPTKDM4EMEN1ALDH1A1TP53
SCHEMBL5779107 0.69 CA12 (0.50) SUCNR1MAPTMEN1ALDH1A1KMT2A
SCHEMBL5778528 0.69 ALB (0.56) SNCAMAPTKDM4EMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1652839-A2 Drug efflux pump inhibitor DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2006-05-03 EP disclosed
EP-1227084-B1 DRUG DISCHARGE PUMP INHIBITORS TRINE PHARMACEUTICALS INC (US) 2005-12-14 EP disclosed
EP-1227084-A1 DRUG DISCHARGE PUMP INHIBITORS Microcide Pharmaceuticals, Inc. (US) 2002-07-31 EP disclosed