SCHEMBL5778188

SCHEMBL5778188

COC(=O)c1cc(OCCO)cc(C(=O)Nc2cccc(C=Cc3nc(C(C)C)cs3)c2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALB P02768 2/20 0.52
SNCA P37840 1/20 0.40
TP53 P04637 4/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
NR1H4 Q96RI1 3/20 0.37
MAPT P10636 4/20 0.36
KDM4E B2RXH2 2/20 0.36
RAB9A P51151 2/20 0.36
ATM Q13315 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
ALDH1A1 P00352 1/20 0.36
ADRB1 P08588 1/20 0.36
CYP3A4 P08684 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
HPGD P15428 1/20 0.36
PTGS1 P23219 1/20 0.36
HSD17B10 Q99714 1/20 0.36
THRB P10828 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5776928 0.93 ALB (0.57) ALBSNCATP53SMN1; SMN2NR1H4
SCHEMBL5775504 0.86 ALB (0.49) ALBSNCATP53SMN1; SMN2NR1H4
SCHEMBL5778528 0.85 ALB (0.56) ALBSNCATP53SMN1; SMN2NR1H4
SCHEMBL5778029 0.79 ALB (0.51) ALBTP53SMN1; SMN2MAPTRAB9A
SCHEMBL5778350 0.77 ALB (0.57) ALBSNCATP53SMN1; SMN2MAPT
SCHEMBL5776526 0.76 SNCA (0.39) ALBSNCATP53SMN1; SMN2NR1H4
SCHEMBL5774563 0.76 ALB (0.69) ALBSNCATP53SMN1; SMN2MAPT
SCHEMBL5778781 0.74 ALB (0.55) ALBSMN1; SMN2MAPTRAB9AMEN1
SCHEMBL5779049 0.74 ALB (0.55) ALBSNCATP53SMN1; SMN2MAPT
SCHEMBL5779175 0.73 ALB (0.55) ALBSNCATP53SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1652839-A2 Drug efflux pump inhibitor DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2006-05-03 EP disclosed
EP-1227084-B1 DRUG DISCHARGE PUMP INHIBITORS TRINE PHARMACEUTICALS INC (US) 2005-12-14 EP disclosed
EP-1227084-A1 DRUG DISCHARGE PUMP INHIBITORS Microcide Pharmaceuticals, Inc. (US) 2002-07-31 EP disclosed