SCHEMBL5776544

SCHEMBL5776544

O=c1[c][c][nH]c2ccccc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.41
ALDH1A1 P00352 6/20 0.41
LMNA P02545 2/20 0.41
GAA P10253 2/20 0.41
HPGD P15428 2/20 0.41
HTT P42858 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
GLA P06280 1/20 0.41
ATM Q13315 1/20 0.41
ALOX5 P09917 2/20 0.40
CYP1A2 P05177 4/20 0.39
PARP1 P09874 2/20 0.39
GPR3 P46089 2/20 0.39
HSD17B10 Q99714 2/20 0.39
TNKS2 Q9H2K2 2/20 0.39
MEN1 O00255 1/20 0.39
TNKS O95271 1/20 0.39
BLM P54132 1/20 0.39
PMP22 Q01453 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15616167 0.74 KDM4E (0.41) KDM4EALDH1A1LMNAGAAHPGD
SCHEMBL223036 0.67 GAA (0.44) KDM4EALDH1A1LMNAGAAHPGD
SCHEMBL3353907 0.65 ALDH1A1 (0.41) KDM4EALDH1A1LMNAGAAHPGD
SCHEMBL555502 0.64 CYP1A2 (0.44) KDM4EALDH1A1LMNAGAAHPGD
SCHEMBL2987901 0.64 ALDH1A1 (0.40) KDM4EALDH1A1LMNAGAAHPGD
SCHEMBL3463581 0.63 KDM4E (0.48) KDM4EALDH1A1LMNAGAAHPGD
SCHEMBL2988035 0.60 CYP2A6 (0.42) KDM4EALDH1A1LMNAGAAHPGD
SCHEMBL1639050 0.59 ALDH1A1 (0.40) KDM4EALDH1A1LMNAGAAHPGD
SCHEMBL3849040 0.59 ALDH1A1 (0.40) KDM4EALDH1A1LMNAGAAHPGD
SCHEMBL570354 0.59 ALDH1A1 (0.40) KDM4EALDH1A1LMNAGAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1652839-A2 Drug efflux pump inhibitor DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2006-05-03 EP claimed
EP-1227084-B1 DRUG DISCHARGE PUMP INHIBITORS TRINE PHARMACEUTICALS INC (US) 2005-12-14 EP claimed
EP-1227084-A1 DRUG DISCHARGE PUMP INHIBITORS Microcide Pharmaceuticals, Inc. (US) 2002-07-31 EP claimed
EP-1652839-A2 Drug efflux pump inhibitor DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2006-05-03 EP disclosed
EP-1227084-B1 DRUG DISCHARGE PUMP INHIBITORS TRINE PHARMACEUTICALS INC (US) 2005-12-14 EP disclosed
EP-1227084-A1 DRUG DISCHARGE PUMP INHIBITORS Microcide Pharmaceuticals, Inc. (US) 2002-07-31 EP disclosed