SCHEMBL5777963

SCHEMBL5777963

Cc1nccn1-c1nc(NCCc2ccc3c(c2)OCO3)c2c3c(sc2n1)CCCC3

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.46
ALDH1A1 P00352 5/20 0.46
ALOX15 P16050 3/20 0.46
LMNA P02545 3/20 0.46
USP2 O75604 2/20 0.46
HTT P42858 6/20 0.45
SMN1; SMN2 Q16637 4/20 0.45
MAPT P10636 6/20 0.44
HSD17B10 Q99714 4/20 0.44
GAA P10253 3/20 0.44
HPGD P15428 3/20 0.44
MAPK1 P28482 3/20 0.44
GLA P06280 2/20 0.44
ATM Q13315 2/20 0.44
NPSR1 Q6W5P4 2/20 0.44
POLB P06746 1/20 0.44
RAD52 P43351 1/20 0.44
PAX8 Q06710 1/20 0.44
TSHR P16473 1/20 0.44
PRKCI P41743 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5780791 0.92 HTT (0.48) KDM4EALDH1A1ALOX15LMNAUSP2
SCHEMBL5781706 0.87 HTT (0.48) KDM4EALDH1A1ALOX15LMNAUSP2
SCHEMBL5124186 0.87 SMN1; SMN2 (0.41) KDM4EALDH1A1LMNAHTTSMN1; SMN2
SCHEMBL5122439 0.85 PDE5A (0.39) KDM4EALDH1A1LMNAHTTSMN1; SMN2
SCHEMBL5122226 0.85 BCDIN3D (0.39) ALDH1A1HTTSMN1; SMN2MAPTNPSR1
SCHEMBL5798539 0.84 NOS2 (0.49) KDM4EALDH1A1ALOX15LMNAUSP2
SCHEMBL5781513 0.84 ALDH1A1 (0.44) KDM4EALDH1A1ALOX15LMNAUSP2
SCHEMBL5130564 0.82 BCDIN3D (0.43) KDM4EALDH1A1SMN1; SMN2HSD17B10MAPK1
SCHEMBL5124067 0.81 BCDIN3D (0.42) KDM4EALDH1A1LMNASMN1; SMN2MAPK1
SCHEMBL5123608 0.81 BCDIN3D (0.42) KDM4EALDH1A1HSD17B10TSHRPRKCI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1685136-A1 USE OF THIENOPYRIMIDINES MERCK PATENT GmbH (DE) 2006-08-02 EP disclosed
WO-2005047292-A1 USE OF THIENOPYRIMIDINES MERCK PATENT GMBH (DE) 2005-05-26 WO disclosed
US-6432950-B1 ANTICANCER AGENTS; KILLING CANCER CELLS CELL PATHWAYS 2002-08-13 US disclosed
US-6133271-A Method for inhibiting neoplastic cells and related conditions by exposure thienopyrimidine derivatives CELL PATHWAYS, INC. (US) 2000-10-17 US disclosed
US-6110920-A TREATMENT OF CARDIOVASCULAR DISORDERS AND IMPOTENCY MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-08-29 US disclosed
EP-0920431-A1 THIENOPYRIMIDINES MERCK PATENT GmbH (DE) 1999-06-09 EP disclosed
WO-1998006722-A1 THIENOPYRIMIDINES MERCK PATENT GMBH (DE) 1998-02-19 WO disclosed