SCHEMBL5778103

SCHEMBL5778103

COc1ccc2ncc(Cl)c(N3CCN(CCNC(=O)CF)CC3)c2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.48
NPSR1 Q6W5P4 2/20 0.48
LMNA P02545 1/20 0.48
MTNR1A P48039 1/20 0.48
MTNR1B P49286 1/20 0.48
POLB P06746 1/20 0.47
DRD4 P21917 5/20 0.46
DRD2 P14416 2/20 0.44
FAAH O00519 1/20 0.43
ACHE P22303 1/20 0.43
HTR1A P08908 2/20 0.43
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
MAPT P10636 2/20 0.43
KDM4E B2RXH2 1/20 0.43
HPGD P15428 1/20 0.43
MAPK1 P28482 1/20 0.43
HSD17B10 Q99714 1/20 0.43
MELK Q14680 1/20 0.43
CYP2D6 P10635 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4063953 0.88 ALDH1A1 (0.47) ALDH1A1NPSR1LMNAMTNR1AMTNR1B
SCHEMBL5778107 0.81 ALDH1A1 (0.49) ALDH1A1NPSR1LMNAMTNR1BPOLB
SCHEMBL4071728 0.80 ALDH1A1 (0.48) ALDH1A1NPSR1LMNAPOLBMAPT
SCHEMBL4068347 0.75 POLB (0.43) ALDH1A1LMNAMTNR1AMTNR1BPOLB
SCHEMBL4064313 0.74 KCNH2 (0.53)
SCHEMBL4069719 0.73 SUV39H2 (0.48) ALDH1A1NPSR1LMNAMTNR1BACHE
SCHEMBL4068253 0.71 KCNH2 (0.48) ALDH1A1NPSR1LMNA
SCHEMBL4066048 0.71 KCNH2 (0.57)
SCHEMBL4064039 0.70 NCF1 (0.53) ALDH1A1MTNR1AMTNR1BDRD4DRD2
SCHEMBL4068344 0.70 KCNH2 (0.42) POLBDRD4DRD2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1605938-A4 ANTIBACTERIAL AGENTS GLAXO GROUP LTD (GB) 2006-11-22 EP disclosed
EP-1605938-A2 ANTIBACTERIAL AGENTS GLAXO GROUP LIMITED (GB) 2005-12-21 EP disclosed
WO-2004087145-A2 ANTIBACTERIAL AGENTS GLAXO GROUP LIMITED (GB) 2004-10-14 WO disclosed