SCHEMBL5778233

SCHEMBL5778233

CCN(Cc1ccccc1)C(=O)c1cnc(Nc2ccccc2Cl)nc1C(F)(F)F

nearest known ligand 0.66

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 14/20 0.66
ATF1 P18846 1/20 0.48
NFKB1 P19838 1/20 0.48
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
ULK1 O75385 1/20 0.42
SIRT5 Q9NXA8 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5778821 0.89 CNR2 (0.68) CNR2ATF1NFKB1CYP1A2CYP2C9
SCHEMBL5779936 0.84 CNR2 (0.67) CNR2CYP1A2CYP2C9
SCHEMBL5079708 0.82 CNR2 (0.59) CNR2ATF1NFKB1CYP1A2CYP2C9
SCHEMBL27694711 0.80 CNR2 (0.72) CNR2CYP1A2CYP2C9ULK1SIRT5
SCHEMBL5780552 0.80 CNR2 (0.56) CNR2ATF1NFKB1CYP1A2CYP2C9
SCHEMBL5782167 0.80 CNR2 (0.56) CNR2ATF1NFKB1CYP1A2CYP2C9
SCHEMBL5780688 0.79 CNR2 (1.00) CNR2CYP1A2CYP2C9SIRT5
SCHEMBL5077147 0.79 CNR2 (0.55) CNR2ATF1NFKB1CYP1A2CYP2C9
SCHEMBL5780970 0.76 CNR2 (0.70) CNR2ATF1NFKB1
SCHEMBL5780255 0.75 CNR2 (0.68) CNR2ATF1NFKB1CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1736470-A2 Pyrimidine derivatives as CB2 cannabinoid receptor modulators GLAXO GROUP LIMITED (GB) 2006-12-27 EP disclosed