SCHEMBL5778272

SCHEMBL5778272

O=C(/C=C/c1cccc([N+](=O)[O-])c1)Nc1cccnc1Cl

nearest known ligand 0.72

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.67
NPC1 O15118 4/20 0.67
ALDH1A1 P00352 2/20 0.67
MEN1 O00255 3/20 0.64
KMT2A Q03164 3/20 0.64
TRPV1 Q8NER1 4/20 0.62
SMN1; SMN2 Q16637 3/20 0.58
HTT P42858 2/20 0.58
SNCA P37840 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5779943 1.00 RAB9A (0.67) RAB9ANPC1ALDH1A1MEN1KMT2A
SCHEMBL3273795 0.79 TRPV1 (0.70) RAB9ANPC1ALDH1A1MEN1KMT2A
SCHEMBL3273786 0.79 TRPV1 (0.70) RAB9ANPC1ALDH1A1MEN1KMT2A
SCHEMBL6791019 0.78 ALDH1A1 (0.80) RAB9ANPC1ALDH1A1MEN1KMT2A
SCHEMBL6791025 0.78 ALDH1A1 (0.80) RAB9ANPC1ALDH1A1MEN1KMT2A
SCHEMBL8641059 0.77 SMN1; SMN2 (0.72) RAB9ANPC1ALDH1A1MEN1KMT2A
SCHEMBL8641053 0.77 SMN1; SMN2 (0.72) RAB9ANPC1ALDH1A1MEN1KMT2A
SCHEMBL1424978 0.77 TRPV1 (0.63) RAB9ANPC1ALDH1A1MEN1KMT2A
SCHEMBL1424974 0.77 TRPV1 (0.63) RAB9ANPC1ALDH1A1MEN1KMT2A
SCHEMBL8065999 0.77 TRPV1 (0.67) RAB9ANPC1ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1652839-A2 Drug efflux pump inhibitor DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2006-05-03 EP disclosed
EP-1227084-B1 DRUG DISCHARGE PUMP INHIBITORS TRINE PHARMACEUTICALS INC (US) 2005-12-14 EP disclosed
EP-1227084-A1 DRUG DISCHARGE PUMP INHIBITORS Microcide Pharmaceuticals, Inc. (US) 2002-07-31 EP disclosed