SCHEMBL5778340

SCHEMBL5778340

O=C(Nc1ccncc1)C1CCN(C(=O)OCc2ccccc2)C(I)C1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
GRIN2B Q13224 1/20 0.52
ENPP2 Q13822 1/20 0.51
POLB P06746 1/20 0.50
F10 P00742 1/20 0.48
KDM1A O60341 1/20 0.48
RCOR1 Q9UKL0 1/20 0.48
TDP1 Q9NUW8 1/20 0.47
KDM4E B2RXH2 1/20 0.47
LMNA P02545 1/20 0.47
HSD17B10 Q99714 1/20 0.46
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
NPSR1 Q6W5P4 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2476561 0.83 ENPP2 (0.70) CYP2D6CYP2C9GRIN2BENPP2POLB
SCHEMBL16568979 0.78 ENPP2 (0.63) CYP2D6CYP2C9GRIN2BENPP2F10
SCHEMBL28219844 0.76 SMN1; SMN2 (0.57) NPC1RAB9ASMN1; SMN2NPSR1
SCHEMBL11750711 0.75 ENPP2 (0.78) CYP2D6CYP2C9GRIN2BENPP2LMNA
SCHEMBL13588931 0.74 KDM4E (0.69) CYP2C9KDM1ARCOR1KDM4ELMNA
SCHEMBL4382017 0.74 KDM4E (0.69) CYP2C9KDM1ARCOR1KDM4ELMNA
SCHEMBL5591753 0.73 PREP (0.48) CYP2D6CYP2C9GRIN2BNPC1RAB9A
SCHEMBL7327862 0.72 ALDH1A1 (0.66) CYP2D6CYP2C9GRIN2BPOLBF10
SCHEMBL7327865 0.72 ALDH1A1 (0.66) CYP2D6CYP2C9GRIN2BPOLBF10
SCHEMBL1554194 0.72 TDP1 (0.61) TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1379520-B1 N-SUBSTITUTED NONARYL-HETEROCYCLIC NMDA/NR2B ANTAGONISTS MERCK & CO INC (US) 2006-04-26 EP disclosed