SCHEMBL5778853

SCHEMBL5778853

O=[N+]([O-])c1cccc(CNc2nc(-c3cnccn3)nc3sc4c(c23)CCCC4)c1

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.47
KDM4E B2RXH2 1/20 0.46
HTT P42858 1/20 0.46
PRKCI P41743 11/20 0.45
RNASEL Q05823 1/20 0.45
PRKCZ Q05513 1/20 0.43
PDE5A O76074 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7512863 0.95 PTGS2 (0.44) PTGS2KDM4EHTTPRKCIRNASEL
SCHEMBL5781685 0.90 MEN1 (0.49) PTGS2HTTPRKCIRNASELPRKCZ
SCHEMBL5780830 0.88 PRKCI (0.53) PTGS2KDM4EHTTPRKCIRNASEL
SCHEMBL5777235 0.87 PRKCI (0.58) PTGS2PRKCIPRKCZ
SCHEMBL5780486 0.85 PDE5A (0.59) PTGS2KDM4EHTTPRKCIPRKCZ
SCHEMBL5802207 0.84 RNASEL (0.49) PTGS2HTTPRKCIRNASELPRKCZ
SCHEMBL5122637 0.83 SMN1; SMN2 (0.46) PRKCIPDE5A
SCHEMBL5802044 0.83 PTGS2 (0.48) PTGS2HTTPRKCIRNASELPRKCZ
SCHEMBL8205517 0.82 PRKCI (0.48) KDM4EHTTPRKCI
SCHEMBL5781751 0.82 RNASEL (0.51) PTGS2KDM4EHTTRNASELPDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1685136-A1 USE OF THIENOPYRIMIDINES MERCK PATENT GmbH (DE) 2006-08-02 EP disclosed
WO-2005047292-A1 USE OF THIENOPYRIMIDINES MERCK PATENT GMBH (DE) 2005-05-26 WO disclosed
US-6110920-A TREATMENT OF CARDIOVASCULAR DISORDERS AND IMPOTENCY MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-08-29 US disclosed