SCHEMBL5779010

SCHEMBL5779010

c1csc(CCNC2CC[N]C2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 1/20 0.42
PDE4A P27815 1/20 0.42
PDE4B Q07343 1/20 0.42
PDE4C Q08493 1/20 0.42
PDE4D Q08499 1/20 0.42
HRH3 Q9Y5N1 2/20 0.40
HSD11B1 P28845 1/20 0.39
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
TAAR1 Q96RJ0 2/20 0.39
GRIN2B Q13224 2/20 0.38
ADAM17 P78536 1/20 0.37
POLB P06746 1/20 0.36
KMT2A Q03164 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
HPGD P15428 1/20 0.36
CYP2C19 P33261 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2094368 0.85 KDM1A (0.46) CHRM3PDE4APDE4BPDE4CPDE4D
SCHEMBL4208468 0.76 SOS1 (0.48) CHRM3PDE4APDE4BPDE4CPDE4D
SCHEMBL2093428 0.75 GRIN2B (0.41) HRH3SMN1; SMN2TAAR1GRIN2BPOLB
SCHEMBL16551625 0.71 GRIN2B (0.63) GRIN2BPOLBKMT2A
SCHEMBL16551698 0.71 GRIN2B (0.63) GRIN2BPOLBKMT2A
SCHEMBL29588794 0.71 GRIN2B (0.63) GRIN2BPOLBKMT2A
SCHEMBL5779830 0.71 MPO (0.45) HRH3TAAR1GRIN2B
SCHEMBL3978945 0.70 SMN1; SMN2 (0.39) CHRM3PDE4APDE4BPDE4CPDE4D
SCHEMBL2030841 0.69 TAAR1 (0.71) HRH3NPC1RAB9ASMN1; SMN2TAAR1
SCHEMBL3034101 0.68 HRH3 (0.43) HRH3GRIN2BPOLBKMT2AKDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1631570-A1 NAPHTHYRIDINE DERIVATIVES AS ANTIBACTERIAL AGENTS Abbott Laboratories (US) 2006-03-08 EP claimed
WO-2004083207-A1 NAPHTHYRIDINE DERIVATIVES AS ANTIBACTERIAL AGENTS ABBOTT LABORATORIES (US) 2004-09-30 WO claimed
EP-1631570-A1 NAPHTHYRIDINE DERIVATIVES AS ANTIBACTERIAL AGENTS Abbott Laboratories (US) 2006-03-08 EP disclosed
WO-2004083207-A1 NAPHTHYRIDINE DERIVATIVES AS ANTIBACTERIAL AGENTS ABBOTT LABORATORIES (US) 2004-09-30 WO disclosed