SCHEMBL5779113

SCHEMBL5779113

CC(NC(=O)O)c1csc(C=NNc2ccc(-c3cnco3)cc2)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 1/20 0.40
NPC1 O15118 5/20 0.39
RAB9A P51151 4/20 0.39
PKM P14618 3/20 0.39
KDM4E B2RXH2 3/20 0.39
LMNA P02545 2/20 0.39
ALDH1A1 P00352 2/20 0.39
IMPDH2 P12268 2/20 0.38
IMPDH1 P20839 1/20 0.38
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38
SYK P43405 1/20 0.36
ACACB O00763 1/20 0.36
POLB P06746 1/20 0.35
PORCN Q9H237 1/20 0.35
JAK3 P52333 1/20 0.35
MAPK1 P28482 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
HTT P42858 1/20 0.34
GAA P10253 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5777358 0.86 AAK1 (0.36) AAK1IMPDH2IMPDH1
SCHEMBL5780662 0.84 CDK4 (0.41) AAK1NPC1RAB9APKMKDM4E
SCHEMBL5912676 0.83 IMPDH2 (0.39) AAK1NPC1RAB9APKMKDM4E
SCHEMBL5774837 0.77 IMPDH2 (0.39) AAK1NPC1RAB9APKMKDM4E
SCHEMBL5780289 0.76 IMPDH2 (0.38) AAK1NPC1RAB9APKMKDM4E
SCHEMBL5779104 0.75 AAK1 (0.38) AAK1NPC1RAB9APKMKDM4E
SCHEMBL5775263 0.75 CDK4 (0.40) AAK1NPC1RAB9APKMKDM4E
SCHEMBL5775549 0.71 IMPDH2 (0.40) AAK1NPC1RAB9APKMKDM4E
SCHEMBL5912811 0.71 IMPDH2 (0.40) AAK1NPC1RAB9APKMKDM4E
SCHEMBL5778654 0.70 CDK4 (0.40) AAK1IMPDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1612204-A1 HYDRAZONE DERIVATIVE DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2006-01-04 EP disclosed