SCHEMBL5779104

SCHEMBL5779104

CC(NC(=O)O)c1csc(/C(=N\N)c2ccc(-c3cnco3)cc2)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 3/20 0.38
PKM P14618 3/20 0.38
NPC1 O15118 3/20 0.38
KDM4E B2RXH2 2/20 0.38
LMNA P02545 2/20 0.38
RAB9A P51151 2/20 0.38
ALDH1A1 P00352 1/20 0.38
ACACB O00763 1/20 0.37
SYK P43405 1/20 0.35
IMPDH2 P12268 2/20 0.35
IMPDH1 P20839 1/20 0.34
HTT P42858 1/20 0.34
MYC P01106 1/20 0.34
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
GPR119 Q8TDV5 2/20 0.33
POLB P06746 1/20 0.33
HDAC3 O15379 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5777356 0.86 AAK1 (0.35) AAK1IMPDH2IMPDH1
SCHEMBL5912671 0.82 IMPDH2 (0.34) AAK1PKMNPC1KDM4ELMNA
SCHEMBL5774833 0.76 GPR119 (0.36) AAK1PKMNPC1KDM4ELMNA
SCHEMBL5779113 0.75 AAK1 (0.40) AAK1PKMNPC1KDM4ELMNA
SCHEMBL5775952 0.72 NPC1 (0.49) AAK1PKMNPC1KDM4ELMNA
SCHEMBL5779456 0.68 GPR119 (0.45) AAK1PKMNPC1KDM4ELMNA
SCHEMBL5777062 0.67 NPC1 (0.44) AAK1PKMNPC1KDM4ELMNA
SCHEMBL5776483 0.66 CDK1 (0.49) AAK1PKMNPC1KDM4ELMNA
SCHEMBL5776708 0.65 ROCK2 (0.41) PKMNPC1KDM4ELMNARAB9A
SCHEMBL5778725 0.65 KDM4E (0.48) AAK1PKMNPC1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1612204-A1 HYDRAZONE DERIVATIVE DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2006-01-04 EP disclosed