SCHEMBL577976

SCHEMBL577976

CC(C)c1csc(-c2cccc3n[c]nc(F)c23)n1

nearest known ligand 0.39

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TYK2 P29597 1/20 0.39
CCR4 P51679 1/20 0.33
HAO1 Q9UJM8 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL577981 0.85 TYK2 (0.35) TYK2CCR4HAO1
SCHEMBL577504 0.82 TYK2 (0.34) TYK2CCR4
SCHEMBL577977 0.82 TYK2 (0.42) TYK2CCR4
SCHEMBL577702 0.80 TYK2 (0.34) TYK2CCR4HAO1
SCHEMBL577982 0.78 CCR4 (0.33) TYK2CCR4
SCHEMBL578408 0.77 TYK2 (0.36) TYK2CCR4HAO1
SCHEMBL577505 0.75 ALDH1A1 (0.36) TYK2CCR4
SCHEMBL577093 0.75 TYK2 (0.34) TYK2CCR4
SCHEMBL577638 0.73 TYK2 (0.33) TYK2
SCHEMBL577273 0.73 KDM4E (0.34) TYK2CCR4HAO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417134-A1 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX Pharmaceuticals, Inc. (US) 2012-02-15 EP disclosed
WO-2010118078-A1 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARMACEUTICALS, INC. (US) 2010-10-14 WO disclosed