SCHEMBL577977

SCHEMBL577977

CC(C)c1csc(-c2n[c]nc3cccc(F)c23)n1

nearest known ligand 0.42

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TYK2 P29597 1/20 0.42
CCR4 P51679 1/20 0.33
PARP1 P09874 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL577982 0.86 CCR4 (0.33) TYK2CCR4PARP1
SCHEMBL577505 0.82 ALDH1A1 (0.36) TYK2CCR4
SCHEMBL577976 0.82 TYK2 (0.39) TYK2CCR4
SCHEMBL577639 0.78 APLNR (0.33) TYK2
SCHEMBL577981 0.77 TYK2 (0.35) TYK2CCR4
SCHEMBL577703 0.75 APLNR (0.32)
SCHEMBL577504 0.75 TYK2 (0.34) TYK2CCR4
SCHEMBL23367842 0.74 TYK2 (0.56) TYK2CCR4
SCHEMBL577608 0.74 SLC10A2 (0.35)
SCHEMBL577533 0.73 APLNR (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417134-A1 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX Pharmaceuticals, Inc. (US) 2012-02-15 EP disclosed
WO-2010118078-A1 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARMACEUTICALS, INC. (US) 2010-10-14 WO disclosed