SCHEMBL5780220

SCHEMBL5780220

Cc1ccc2cc(OCCN3CCN(Cc4ccc5c(c4)N(S(C)(=O)=O)CCO5)CC3)ccc2n1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 18/20 0.49
HTR1B P28222 18/20 0.49
HTR1A P08908 16/20 0.49
CYP2C9 P11712 5/20 0.49
CYP1A2 P05177 4/20 0.49
CYP2C19 P33261 3/20 0.47
CYP3A4 P08684 2/20 0.47
CYP2D6 P10635 2/20 0.47
DRD3 P35462 1/20 0.39
KCNH2 Q12809 1/20 0.39
MAOB P27338 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5367054 0.84 HTR1D (0.71) HTR1DHTR1BHTR1ACYP2C9CYP1A2
SCHEMBL5361811 0.83 HTR1D (0.57) HTR1DHTR1BHTR1ACYP2C9CYP1A2
SCHEMBL5369049 0.80 HTR1D (0.51) HTR1DHTR1BHTR1ACYP2C9CYP1A2
SCHEMBL5780146 0.79 HTR1D (0.47) HTR1DHTR1BHTR1ACYP2C9CYP1A2
SCHEMBL5364330 0.77 HTR1D (0.57) HTR1DHTR1BHTR1ACYP2C9CYP1A2
SCHEMBL5364221 0.73 HTR1A (0.72) HTR1DHTR1BHTR1ADRD3
SCHEMBL5369043 0.71 FAAH (0.50) CYP2D6
SCHEMBL5361819 0.71 PDE3B (0.47) CYP2D6
SCHEMBL13185173 0.67 PDE3B (0.51) CYP2C9
SCHEMBL5371636 0.66 PDE3B (0.53) CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1476444-B1 HETEROCYCLIC COMPOUNDS POSSESSING AFFINITY AT 5HT1-TYPE RECEPTORS AND USE THEREOF IN THERAPY GLAXO GROUP LTD (GB) 2006-04-12 EP claimed