SCHEMBL5780334

SCHEMBL5780334

CC(C)(C)NC(=O)N1CC(OC(c2ccccc2)c2ccc(Cl)cc2C(F)(F)F)C1

nearest known ligand 0.50

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 4/20 0.41
CNR2 P34972 3/20 0.41
CYP3A4 P08684 1/20 0.41
CYP3A5 P20815 1/20 0.41
FAAH O00519 10/20 0.41
RORC P51449 1/20 0.40
TACR1 P25103 1/20 0.40
ALDH1A1 P00352 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5800214 0.90 FAAH (0.40) CNR1CNR2FAAHALDH1A1SMN1; SMN2
SCHEMBL5782662 0.89 TACR1 (0.47) CNR1CNR2CYP3A4FAAHRORC
SCHEMBL5804489 0.89 GRIN2B (0.47) CNR1CNR2FAAH
Selonabant SCHEMBL4075847 0.88 CNR1 (0.49) CNR1CNR2FAAH
Selonabant SCHEMBL29482761 0.88 CNR1 (0.49) CNR1CNR2FAAH
Selonabant SCHEMBL4075536 0.88 CNR1 (0.49) CNR1CNR2FAAH
Selonabant SCHEMBL4075537 0.88 CNR1 (0.49) CNR1CNR2FAAH
Selonabant SCHEMBL31259163 0.88 CNR1 (0.49) CNR1CNR2FAAH
SCHEMBL4089353 0.88 RORC (0.44) CNR1CNR2FAAHRORCTACR1
SCHEMBL4084803 0.88 TACR1 (0.45) CNR1CNR2CYP3A4CYP3A5FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1620395-A1 AZETIDINECARBOXAMIDE DERIVATIVES AND THEIR USE IN THE TREATMENT OF CB1 RECEPTOR MEDIATED DISORDERS VERNALIS RESEARCH LIMITED (GB) 2006-02-01 EP disclosed
WO-2004096763-A1 AZETIDINECARBOXAMIDE DERIVATIVES AND THEIR USE IN THE TREATMENT OF CB1 RECEPTOR MEDIATED DISORDERS VERNALIS RESEARCH LIMITED (GB) 2004-11-11 WO disclosed