SCHEMBL5780394

SCHEMBL5780394

CC(C)(C)OC(=O)NC(CS(=O)(=O)CC1(c2cccc3c2oc2ccccc23)C=CC(c2ccccc2)=CC1)C(=O)O

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.35
TSHR P16473 1/20 0.35
EPHX2 P34913 1/20 0.34
ACE P12821 2/20 0.34
CTSS P25774 4/20 0.34
CTSK P43235 3/20 0.34
BCL2 P10415 1/20 0.33
PPARA Q07869 5/20 0.33
PPARG P37231 4/20 0.33
IDO1 P14902 1/20 0.33
MMP13 P45452 2/20 0.33
AKT1 P31749 1/20 0.32
PPARD Q03181 2/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
ATM Q13315 1/20 0.32
CTSL P07711 1/20 0.32
CTSB P07858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5200688 0.86 PPARA (0.42) TSHREPHX2ACECTSSCTSK
SCHEMBL5262506 0.82 EPHX2 (0.33) EPHX2ACECTSSCTSKPPARA
SCHEMBL5781491 0.81 ACE (0.37) ALDH1A1EPHX2ACECTSSCTSK
SCHEMBL5783679 0.73 PPARA (0.41) TSHREPHX2ACECTSSCTSK
SCHEMBL4818610 0.73 PTPN1 (0.42) ALDH1A1TSHREPHX2ACECTSS
SCHEMBL4821211 0.73 PTPN1 (0.42) ALDH1A1TSHREPHX2ACECTSS
SCHEMBL9956802 0.70 CTSS (0.56) EPHX2ACECTSSCTSKPPARA
SCHEMBL5764439 0.70 MAPT (0.33) ALDH1A1
SCHEMBL4824631 0.70 PPARA (0.42) ACECTSSCTSKPPARAPPARG
SCHEMBL5197297 0.69 CTSS (0.36) ALDH1A1TSHREPHX2ACECTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1622886-A2 SUBSTITUTED AMINO CARBOXYLIC ACIDS AS INHIBITORS OF PROTEIN TYROSINE PHOSPHATASE-1B The Institutes for Pharmaceutical Discovery, LLC (US) 2006-02-08 EP disclosed
WO-2004099171-A2 SUBSTITUTED AMINO CARBOXYLIC ACIDS AS INHIBITORS OF PROTEIN TYROSINE PHOSPHATASE-1B THE INSTITUTES FOR PHARMACEUTICAL DISCOVERY, LLC (US) 2004-11-18 WO disclosed