SCHEMBL5780690

SCHEMBL5780690

N#Cc1ccc2c(=O)ccoc2c1

nearest known ligand 0.64

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.64
FTO Q9C0B1 2/20 0.56
CYP2A6 P11509 1/20 0.53
KDM4E B2RXH2 1/20 0.51
MAOA P21397 6/20 0.51
MAOB P27338 6/20 0.51
CA1 P00915 2/20 0.46
CA2 P00918 2/20 0.46
CYP19A1 P11511 3/20 0.45
ROCK2 O75116 1/20 0.45
ROCK1 Q13464 1/20 0.45
TNKS O95271 1/20 0.42
XDH P47989 1/20 0.41
SLC22A12 Q96S37 1/20 0.41
NOS3 P29474 1/20 0.40
NOS1 P29475 1/20 0.40
NOS2 P35228 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30744099 1.00 GRM5 (0.64) GRM5FTOCYP2A6KDM4EMAOA
SCHEMBL20301257 0.86 MAOA (0.62) GRM5FTOCYP2A6KDM4EMAOA
SCHEMBL506960 0.73 CYP2A6 (0.71) CYP2A6KDM4EMAOAMAOBCA1
SCHEMBL28230155 0.73 FTO (0.63) GRM5FTOKDM4EMAOAMAOB
SCHEMBL826634 0.73 CYP2A6 (0.46) GRM5FTOCYP2A6KDM4EMAOA
SCHEMBL3681299 0.72 FTO (0.61) GRM5FTOCYP2A6KDM4EMAOA
SCHEMBL2065762 0.72 FTO (0.61) GRM5FTOCYP2A6KDM4EMAOA
SCHEMBL546240 0.72 FTO (1.00) GRM5FTOCYP2A6KDM4EMAOA
SCHEMBL29799642 0.72 FTO (1.00) GRM5FTOCYP2A6KDM4EMAOA
SCHEMBL903208 0.72 FTO (0.61) GRM5FTOKDM4EMAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1511734-A4 COMPOUNDS, COMPOSITIONS, AND METHODS CYTOKINETICS INC (US) 2006-05-10 EP disclosed
EP-1511734-A2 COMPOUNDS, COMPOSITIONS, AND METHODS Cytokinetics, Inc. (US) 2005-03-09 EP disclosed
WO-2003088903-A2 COMPOUNDS, COMPOSITIONS, AND METHODS CYTOKINETICS, INC. (US) 2003-10-30 WO disclosed