SCHEMBL5780765

SCHEMBL5780765

CC(O)CC(C)(c1cccc(F)c1)C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 4/20 0.39
CETP P11597 2/20 0.36
NR3C1 P04150 1/20 0.34
PGR P06401 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34
PTPN1 P18031 1/20 0.34
KIF11 P52732 1/20 0.34
CHRM3 P20309 1/20 0.34
NR3C2 P08235 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5780276 0.80 HSD11B1 (0.39) KCNN4
SCHEMBL3812826 0.74 NR3C1 (0.41) NR3C1PGRCHRM3NR3C2
SCHEMBL3680226 0.73 CETP (0.46) KCNN4CETPNR3C1PGRGAA
SCHEMBL13251355 0.71 KCNN4 (0.41) KCNN4CETPHTR2AHTR2CHTR2B
SCHEMBL3655404 0.71 NR3C2 (0.49) NR3C1PGRNR3C2
SCHEMBL30467945 0.70 KCNN4 (0.46) KCNN4NR3C1PGRPTPN1KIF11
SCHEMBL25134588 0.69 KCNN4 (0.48) KCNN4PTPN1KIF11CHRM3ALDH1A1
SCHEMBL25134589 0.69 KCNN4 (0.48) KCNN4PTPN1KIF11HDAC3HDAC1
SCHEMBL25502577 0.69 KCNN4 (0.44) KCNN4HTR2AHTR2CHTR2BPTPN1
SCHEMBL24824473 0.68 KCNN4 (0.52) KCNN4PTPN1KIF11CHRM3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1673088-A1 1,1,1- TRIFLUORO-4-PHENYL-4-METHYL-2-(1H-PYRROLO¬2,3-C|PYRIDIN-2-YLMETHYL)PENTAN-2-OL DERIVATIVES AND RELATED COMPOUNDS AS GLUCOCORTICOID LIGANDS FOR THE TREATMENT OF INFLAMMATORY DISEASES AND DIABETES BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2006-06-28 EP disclosed
WO-2005030213-A1 1,1,1-TRIFLUORO-4-PHENYL-4-METHYL-2-(1H-PYRROLO BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2005-04-07 WO disclosed