SCHEMBL5780971

SCHEMBL5780971

COc1ccc(CNc2nc(-c3cccnc3)nc3sc4c(c23)CCCC4)cc1Cl

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.54
ALDH1A1 P00352 2/20 0.54
GAA P10253 1/20 0.54
MAPT P10636 1/20 0.54
NPC1 O15118 1/20 0.52
NFKB1 P19838 1/20 0.52
RAB9A P51151 1/20 0.52
NFKB2 Q00653 1/20 0.52
RELA Q04206 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
PRKCI P41743 14/20 0.51
PTGS2 P35354 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7169369 0.97 KDM4E (0.51) KDM4EALDH1A1GAAMAPTNPC1
SCHEMBL5781064 0.93 KDM4E (0.55) KDM4EALDH1A1GAAMAPTNPC1
SCHEMBL7169927 0.91 KDM4E (0.50) KDM4EALDH1A1GAAMAPTNPC1
SCHEMBL5778475 0.90 PRKCI (0.62) PRKCI
SCHEMBL7197493 0.90 KDM4E (0.44) KDM4EALDH1A1GAAMAPTNPC1
SCHEMBL5777689 0.90 KDM4E (0.58) KDM4EALDH1A1GAAMAPTNPC1
SCHEMBL5780526 0.87 PRKCI (0.49) MAPTSMN1; SMN2PRKCIPTGS2
SCHEMBL7174213 0.87 KDM4E (0.55) KDM4EALDH1A1GAAMAPTNPC1
SCHEMBL7198624 0.86 PRKCI (0.54) KDM4EALDH1A1GAAMAPTPRKCI
SCHEMBL5127640 0.85 PDE5A (0.46) KDM4EALDH1A1MAPTNPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1685136-A1 USE OF THIENOPYRIMIDINES MERCK PATENT GmbH (DE) 2006-08-02 EP disclosed
WO-2005047292-A1 USE OF THIENOPYRIMIDINES MERCK PATENT GMBH (DE) 2005-05-26 WO disclosed
US-6110920-A TREATMENT OF CARDIOVASCULAR DISORDERS AND IMPOTENCY MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-08-29 US disclosed