Predicted protein targets (top 4)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | TSHR | P16473 | 1/20 | 0.35 |
| ▸ | LMNA | P02545 | 1/20 | 0.33 |
| ▸ | KMT2A | Q03164 | 2/20 | 0.32 |
| ▸ | BLM | P54132 | 1/20 | 0.31 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| SCHEMBL5695118 | 0.79 | TSHR (0.35) | TSHRLMNAKMT2ABLM | |
| SCHEMBL1177989 | 0.77 | TSHR (0.34) | TSHRLMNAKMT2ABLM | |
| SCHEMBL8734424 | 0.77 | TSHR (0.35) | TSHRLMNAKMT2ABLM | |
| SCHEMBL11637189 | 0.77 | LMNA (0.33) | TSHRLMNAKMT2A | |
| SCHEMBL3690646 | 0.77 | LMNA (0.35) | TSHRLMNAKMT2A | |
| SCHEMBL9177970 | 0.76 | LMNA (0.38) | LMNA | |
| SCHEMBL4607227 | 0.76 | KMT2A (0.40) | TSHRLMNAKMT2ABLM | |
| SCHEMBL1226609 | 0.75 | TSHR (0.54) | TSHRLMNAKMT2ABLM | |
| SCHEMBL5859538 | 0.74 | TSHR (0.33) | TSHRLMNAKMT2A | |
| SCHEMBL2441909 | 0.74 | KMT2A (0.33) | TSHRKMT2A |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 144 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| CN-118019524-A | Dydrogesterone sustained release pharmaceutical composition | 曼肯制药有限公司 | 2024-05-10 | — | — | CN | claimed |
| US-20240032530-A1 | BLOOD SAMPLER CONTAINING ANTI-PLATELET AGENT AND WATER-SOLUBLE MATRIX MATERIAL | RADIOMETER MEDICAL APS (DK) | 2024-02-01 | — | — | US | claimed |
| EP-4267003-A1 | BLOOD SAMPLER CONTAINING ANTI-PLATELET AGENT AND WATER-SOLUBLE MATRIX MATERIAL | Radiometer Medical ApS (DK) | 2023-11-01 | — | — | EP | claimed |
| US-20230220560-A1 | Aqueous Pickling Compositions and Their Use | CHEMETALL GMBH (DE) | 2023-07-13 | — | — | US | claimed |
| EP-4165231-A1 | AQUEOUS PICKLING COMPOSITIONS AND THEIR USE | Chemetall GmbH (DE) | 2023-04-19 | — | — | EP | claimed |
| WO-2022136545-A1 | BLOOD SAMPLER CONTAINING ANTI-PLATELET AGENT AND WATER-SOLUBLE MATRIX MATERIAL | RADIOMETER MEDICAL APS (DK) | 2022-06-30 | — | — | WO | claimed |
| WO-2021249880-A1 | AQUEOUS PICKLING COMPOSITIONS AND THEIR USE | CHEMETALL GMBH (DE) | 2021-12-16 | — | — | WO | claimed |
| EP-3368084-A1 | PHARMACEUTICAL COMPOSITIONS FOR TRANSMUCOSAL DELIVERY | Solubest Ltd (IL) | 2018-09-05 | — | — | EP | claimed |
| US-20170119660-A1 | PHARMACEUTICAL COMPOSITIONS FOR TRANSMUCOSAL DELIVERY | SOLUBEST LTD (IL) | 2017-05-04 | — | — | US | claimed |
| WO-2017072774-A1 | PHARMACEUTICAL COMPOSITIONS FOR TRANSMUCOSAL DELIVERY | SOLUBEST LTD (IL) | 2017-05-04 | — | — | WO | claimed |
| WO-2010096814-A1 | CONTROLLED-RELEASE COMPOSITIONS COMPRISING A PROTON PUMP INHIBITOR | EURAND, INC. (US) | 2010-08-26 | — | — | WO | claimed |
| WO-2010077927-A1 | COMPOSITIONS COMPRISING MELPERONE AND CONTROLLED-RELEASE DOSAGE FORMS | EURAND, INC. (US) | 2010-07-08 | — | — | WO | claimed |
| EP-2200588-A1 | COMPOSITIONS COMPRISING LIPOPHILIC ACTIVE COMPOUNDS AND METHOD FOR THEIR PREPARATION | Solubest Ltd. (IL) | 2010-06-30 | — | — | EP | claimed |
| US-20100151015-A1 | Compositions Comprising Melperone and Controlled-Release Dosage Forms | APTALIS PHARMATECH, INC. | 2010-06-17 | — | — | US | claimed |
| US-20100151021-A1 | Compositions Comprising Melperone | APTALIS PHARMATECH, INC. | 2010-06-17 | — | — | US | claimed |
| WO-2009040818-A9 | COMPOSITIONS COMPRISING LIPOPHILIC ACTIVE COMPOUNDS AND METHOD FOR THEIR PREPARATION | SOLUBEST LTD (IL) | 2010-05-20 | — | — | WO | claimed |
| WO-2009129282-A1 | COMPOSITIONS COMPRISING WEAKLY BASIC DRUGS AND CONTROLLED-RELEASE DOSAGE FORMS | EURAND INC (US) | 2009-10-22 | — | — | WO | claimed |
| US-20090258066-A1 | COMPOSITIONS COMPRISING WEAKLY BASIC DRUGS AND CONTROLLED-RELEASE DOSAGE FORMS | ADARE PHARMACEUTICALS USA, INC. | 2009-10-15 | — | — | US | claimed |
| US-20090098200-A1 | COMPOSITIONS COMPRISING LIPOPHILIC ACTIVE COMPOUNDS AND METHOD FOR THEIR PREPARATION | SOLUBEST LTD. (IL) | 2009-04-16 | — | — | US | claimed |
| WO-2009040818-A1 | COMPOSITIONS COMPRISING LIPOPHILIC ACTIVE COMPOUNDS AND METHOD FOR THEIR PREPARATION | SOLUBEST LTD (IL) | 2009-04-02 | — | — | WO | claimed |