SCHEMBL5783192

SCHEMBL5783192

N#CC[C@H]1CCC[C@@H](CN2C(=O)c3cccc(NC(=O)C4=CC(Cl)=CCC4=S)c3C2=O)C1

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.38
RPS6KA2 Q15349 2/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP1B1 Q16678 1/20 0.31
TRPA1 O75762 1/20 0.30
NR1I2 O75469 1/20 0.30
UGCG Q16739 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6214525 0.88 ACHE (0.44) ACHERPS6KA2KDM4EALDH1A1NR1I2
SCHEMBL5784229 0.86 ACHE (0.38) ACHERPS6KA2KDM4EALDH1A1CYP1B1
SCHEMBL5784019 0.85
SCHEMBL5784447 0.84 ACHE (0.41) ACHERPS6KA2KDM4EALDH1A1CYP1B1
SCHEMBL6220121 0.84 ACHE (0.41) ACHERPS6KA2KDM4EALDH1A1NR1I2
SCHEMBL5783534 0.82 HDAC1 (0.40) ACHERPS6KA2KDM4EALDH1A1
SCHEMBL6218958 0.81 ACHE (0.55) ACHERPS6KA2
SCHEMBL5781219 0.81 ACHE (0.39) ACHERPS6KA2KDM4EALDH1A1
SCHEMBL5803057 0.80 ACHE (0.39) ACHERPS6KA2KDM4EALDH1A1
SCHEMBL5783190 0.80 ACHE (0.40) ACHERPS6KA2KDM4EALDH1A1CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1408962-B1 SUBSTITUTED ISOINDOLES AND THE USE THEREOF BAYER HEALTHCARE AG (DE) 2006-03-15 EP disclosed