SCHEMBL5783709

SCHEMBL5783709

NC(=O)CC(NS(=O)(=O)c1cccc2ccccc12)c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC1A3 P43003 1/20 0.56
SLC1A2 P43004 1/20 0.56
SLC1A1 P43005 1/20 0.56
KCNA5 P22460 1/20 0.51
F2 P00734 5/20 0.49
PRSS1 P07477 2/20 0.49
PRSS2 P07478 2/20 0.49
PRSS3 P35030 2/20 0.49
CASP1 P29466 1/20 0.47
ATM Q13315 2/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
TSHR P16473 1/20 0.46
EEF2K O00418 3/20 0.44
ALDH1A1 P00352 2/20 0.43
F10 P00742 2/20 0.43
KDM4E B2RXH2 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2202179 0.90 ATM (0.58) SLC1A3SLC1A2SLC1A1KCNA5F2
SCHEMBL2204265 0.85 KCNA5 (0.52) SLC1A3SLC1A2SLC1A1KCNA5F2
SCHEMBL6496422 0.83 SLC1A3 (0.61) SLC1A3SLC1A2SLC1A1F2PRSS1
SCHEMBL27580332 0.83 SLC1A3 (0.61) SLC1A3SLC1A2SLC1A1F2PRSS1
SCHEMBL27410492 0.80 SLC1A3 (0.53) SLC1A3SLC1A2SLC1A1F2PRSS1
SCHEMBL5674838 0.78 ATM (0.49) ATML3MBTL1EEF2KALDH1A1CYP1A2
SCHEMBL13985124 0.77 SLC1A3 (0.56) SLC1A3SLC1A2SLC1A1F2PRSS1
SCHEMBL6652039 0.77 SLC1A3 (0.56) SLC1A3SLC1A2SLC1A1F2PRSS1
SCHEMBL2693257 0.77 SLC1A3 (0.63) SLC1A3SLC1A2SLC1A1KCNA5F2
SCHEMBL7785619 0.76 ATM (0.42) SLC1A3SLC1A2SLC1A1KCNA5F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1631542-A1 BICYCLIC COMPOUNDS HAVING BRADYKININ RECEPTORS AFFINITY AND PHARMACEUTICAL COMPOSITIONS THEREOF Amgen, Inc. (US) 2006-03-08 EP disclosed
WO-2004092116-A1 BICYCLIC COMPOUNDS HAVING BRADYKININ RECEPTORS AFFINITY AND PHARMACEUTICAL COMPOSITIONS THEREOF AMGEN, INC. (US) 2004-10-28 WO disclosed