SCHEMBL5788904

SCHEMBL5788904

CC(C)(C)OC(=O)N1CCC(=O)CC1.CC(C)(C)OC(=O)N1CCC(CN)CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.48
PKM P14618 1/20 0.48
MAPT P10636 2/20 0.46
THRB P10828 1/20 0.46
HPGD P15428 1/20 0.46
DDB1 Q16531 1/20 0.45
CRBN Q96SW2 1/20 0.45
GPR119 Q8TDV5 7/20 0.45
FAAH O00519 1/20 0.44
RECQL P46063 1/20 0.44
EPHX1 P07099 1/20 0.44
NPC1 O15118 1/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPK1 P28482 1/20 0.43
HTT P42858 1/20 0.43
RAB9A P51151 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
PTPN2 P17706 1/20 0.43
PTPN1 P18031 1/20 0.43
PTPN6 P29350 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL103083 0.90 HPGD (0.54) KDM4EPKMMAPTTHRBHPGD
Hydrochloric Acid SCHEMBL735395 0.88 HPGD (0.53) KDM4EPKMMAPTTHRBHPGD
SCHEMBL17221591 0.84 HPGD (0.56) KDM4EPKMMAPTHPGDGPR119
SCHEMBL7819063 0.84 MAPT (0.52) KDM4EMAPTTHRBHPGDDDB1
SCHEMBL27669441 0.83 USP2 (0.56) KDM4EMAPTTHRBHPGDDDB1
SCHEMBL31028 0.83 USP2 (0.56) KDM4EMAPTTHRBHPGDDDB1
SCHEMBL8152888 0.82 MAPT (0.50) KDM4EMAPTTHRBHPGDDDB1
SCHEMBL4508565 0.82 GPR119 (0.48) KDM4EPKMMAPTTHRBGPR119
Ammonia Solution, Strong SCHEMBL27841683 0.82 USP2 (0.55) KDM4EMAPTTHRBHPGDDDB1
SCHEMBL8993970 0.82 HPGD (0.47) KDM4EPKMMAPTTHRBHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1644356-A1 SUBSTITUTED 4-AMINO-1-BENZYLPIPERIDINE COMPOUNDS Theravance, Inc. (US) 2006-04-12 EP disclosed
WO-2005007645-A1 SUBSTITUTED 4-AMINO-1-BENZYLPIPERIDINE COMPOUNDS THERAVANCE, INC. (US) 2005-01-27 WO disclosed