SCHEMBL5789282

SCHEMBL5789282

N#Cc1ccc(O)c(Cl)c1Cl

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.48
MAPK1 P28482 1/20 0.48
AR P10275 11/20 0.46
ESR1 P03372 4/20 0.45
ESR2 Q92731 4/20 0.45
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
HTR2B P41595 1/20 0.40
TRPV4 Q9HBA0 1/20 0.39
UPP1 Q16831 1/20 0.38
CXCR1 P25024 1/20 0.37
CXCR2 P25025 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31621318 0.84 AR (0.50) CYP3A4MAPK1ARHTR2AHTR2C
SCHEMBL10733139 0.84 AR (0.50) CYP3A4MAPK1ARHTR2AHTR2C
SCHEMBL8996023 0.84 CXCR1 (0.43) CYP3A4MAPK1ARESR1ESR2
SCHEMBL1930255 0.80 AR (0.53) AR
SCHEMBL2518863 0.79 TSHR (0.50) CYP3A4MAPK1ARESR1ESR2
SCHEMBL24636778 0.76 AR (0.43) CYP3A4MAPK1ARESR1ESR2
SCHEMBL68064 0.76 CYP3A4 (0.75) CYP3A4MAPK1ESR1ESR2
SCHEMBL7743436 0.76 CYP3A4 (0.75) CYP3A4MAPK1ESR1ESR2
SCHEMBL31392414 0.76 CYP3A4 (0.75) CYP3A4MAPK1ESR1ESR2
SCHEMBL2869595 0.75 TRPV4 (0.46) CYP3A4MAPK1ARHTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006009937-A2 NOVEL ESTERS AS USEFUL BROAD SPECTRUM HERBICIDAL COMPOUNDS CORET JOEL MARCEL (US) 2006-01-26 WO claimed
CN-110997838-B Silicone-polyether copolymers, sealants including silicone-polyether copolymers, and related methods 美国陶氏有机硅公司 2021-10-01 CN disclosed
EP-1126833-A4 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES INC (US) 2004-09-08 EP disclosed
EP-1126833-A2 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES, INC. (US) 2001-08-29 EP disclosed
WO-2000025768-A1 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES, INC. (US) 2000-05-11 WO disclosed
US-5643929-A TREATMENT OF PICORNAVIRAL OR RHINOVIRUS AND CHEMICAL INTERMEDIATES SANOFI WINTHROP, INC. (US) 1997-07-01 US disclosed
US-4348401-A ANTIHISTAMINIC, ANTIEDEMIC, ANTIPHLOGISTIC BOEHRINGER MANNHEIM GMBH (DE) 1982-09-07 US disclosed