SCHEMBL5789313

SCHEMBL5789313

Cc1ccccc1N(C)c1ccc(CNC(=O)c2cccn(-c3cc(C(F)(F)F)ccc3C)c2=O)cc1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ELANE P08246 5/20 0.41
KDM4E B2RXH2 5/20 0.41
ALDH1A1 P00352 5/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
GAA P10253 1/20 0.40
TACR1 P25103 1/20 0.39
HTT P42858 1/20 0.38
SCD O00767 1/20 0.38
UGCG Q16739 1/20 0.38
LSS P48449 1/20 0.38
DRD2 P14416 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5758984 0.90 KDM4E (0.45) ELANEKDM4EALDH1A1SMN1; SMN2GAA
SCHEMBL6215080 0.84 RECQL (0.44) ELANEKDM4EALDH1A1SMN1; SMN2LSS
SCHEMBL5755996 0.84 CCR1 (0.48) ELANEKDM4EALDH1A1SMN1; SMN2HTT
SCHEMBL5759223 0.83 RECQL (0.48) ELANEKDM4EALDH1A1SMN1; SMN2
SCHEMBL5758300 0.78 ALDH1A1 (0.50) KDM4EALDH1A1SMN1; SMN2HTT
SCHEMBL5755639 0.72 CYP1A2 (0.48) KDM4EALDH1A1SMN1; SMN2HTT
SCHEMBL5755268 0.70 ALDH1A1 (0.48) KDM4EALDH1A1HTT
SCHEMBL5757140 0.70 HPGD (0.54) KDM4EALDH1A1SMN1; SMN2
SCHEMBL27644620 0.68 TP53 (0.41) KDM4EALDH1A1HTT
SCHEMBL5757397 0.66 ELANE (0.75) ELANEKDM4EALDH1A1SMN1; SMN2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562902-B1 2-PYRIDONE DERIVATIVES AS INHIBITORS OF NEUTROPHILE ELASTASE ASTRAZENECA AB (SE) 2006-05-03 EP disclosed