SCHEMBL5789705

SCHEMBL5789705

NC(N)CCCc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.54
GRIK1 P39086 1/20 0.53
MAOB P27338 2/20 0.52
HTR2A P28223 2/20 0.52
IDO1 P14902 1/20 0.50
SIGMAR1 Q99720 1/20 0.48
CYP2A6 P11509 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
TAAR1 Q96RJ0 1/20 0.48
LOXL2 Q9Y4K0 1/20 0.48
ANPEP P15144 2/20 0.47
ERAP1 Q9NZ08 2/20 0.47
ERAP2 Q6P179 1/20 0.47
HTR3A P46098 1/20 0.47
AOC3 Q16853 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10535805 0.98 MAOB (0.54) MAOAGRIK1MAOBHTR2AIDO1
SCHEMBL3266047 0.86 S1PR2 (0.59) MAOAGRIK1MAOBHTR2AIDO1
SCHEMBL829786 0.85 ANPEP (0.55) MAOAMAOBHTR2AIDO1SIGMAR1
Hydrochloric Acid SCHEMBL1979100 0.84 S1PR2 (0.57) MAOAGRIK1MAOBHTR2AIDO1
Bromide SCHEMBL10928757 0.83 SIGMAR1 (0.50) MAOAMAOBHTR2AIDO1SIGMAR1
SCHEMBL29017813 0.82 HTR2A (0.57) MAOAHTR2ASIGMAR1
SCHEMBL3712834 0.82 SLC6A2 (0.56) MAOAGRIK1MAOBHTR2ASIGMAR1
SCHEMBL29029777 0.82 MAOA (0.50) MAOAGRIK1MAOBHTR2AIDO1
SCHEMBL14544283 0.82 GRIK1 (0.54) MAOAGRIK1MAOBHTR2AIDO1
SCHEMBL456442 0.82 GRIK1 (0.54) MAOAGRIK1MAOBHTR2AIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633348-A1 4- BROMO - 5 - (2- CHLORO - BENZOYLAMINO) - 1H - PYRAZOLE - 3 - CARBOXYLIC ACID AMIDE DERIVATIVES AND RELATED COMPOUNDS AS BRADYKININ B sb 1 /sb RECEPTOR ANTAGONISTS FOR THE TREATMENT OF INFLAMMATORY DISEASES Elan Pharmaceuticals, Inc. (US) 2006-03-15 EP claimed
WO-2004098589-A1 4- BROMO - 5 - (2- CHLORO - BENZOYLAMINO) - 1H - PYRAZOLE - 3 - CARBOXYLIC ACID AMIDE DERIVATIVES AND RELATED COMPOUNDS AS BRADYKININ B1 RECEPTOR ANTAGONISTS FOR THE TREATMENT OF INFLAMMATORY DISEASES ELAN PHARMACEUTICALS, INC. (US) 2004-11-18 WO claimed