SCHEMBL5789808

SCHEMBL5789808

CC1CN(Cc2ccc(C#N)c(NC(c3ccccc3)c3ccccc3)c2)C(=O)[C@H](C)N1C(=O)O

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CACNA1G O43497 15/20 0.36
CACNA1H O95180 15/20 0.36
CACNA1I Q9P0X4 15/20 0.36
CYP2D6 P10635 1/20 0.35
OPRK1 P41145 1/20 0.35
S1PR3 Q99500 1/20 0.35
CHRM2 P08172 2/20 0.34
CHRM1 P11229 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP3A4 P08684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4388057 0.89 CACNA1G (0.49) CACNA1GCACNA1HCACNA1ICYP2D6CHRM2
SCHEMBL7375950 0.89 CACNA1G (0.49) CACNA1GCACNA1HCACNA1ICYP2D6CHRM2
SCHEMBL4399774 0.71 CACNA1G (0.54) CACNA1GCACNA1HCACNA1ICHRM2CHRM1
SCHEMBL4399779 0.71 CACNA1G (0.54) CACNA1GCACNA1HCACNA1ICHRM2CHRM1
SCHEMBL18425663 0.61 CACNA1G (0.50) CACNA1GCACNA1HCACNA1I
SCHEMBL20241880 0.61 KDM4E (0.46) ALDH1A1
SCHEMBL22506821 0.61 CACNA1G (0.50) CACNA1GCACNA1HCACNA1I
SCHEMBL20241734 0.60 HTR6 (0.64)
SCHEMBL21378870 0.60 HTR6 (0.48) ALDH1A1
SCHEMBL20242020 0.59 HTR6 (0.50) CYP2D6ALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051176-B1 SUBSTITUTED OXOAZAHETEROCYCLYL FACTOR Xa INHIBITORS AVENTIS PHARMA INC (US) 2006-11-22 EP disclosed