SCHEMBL5790355

SCHEMBL5790355

S=C=NCc1ccc(CCl)cc1

nearest known ligand 0.63

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MIF P14174 14/20 0.63
TRPA1 O75762 3/20 0.63
ALDH1A1 P00352 1/20 0.61
CYP3A4 P08684 1/20 0.61
HPGD P15428 1/20 0.61
CYP2E1 P05181 1/20 0.38
CYP2A6 P11509 1/20 0.38
HIF1A Q16665 1/20 0.38
CYP2A13 Q16696 1/20 0.38
EPAS1 Q99814 1/20 0.38
P2RY6 Q15077 1/20 0.35
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
NAAA Q02083 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2141861 0.88 MIF (0.77) MIFTRPA1ALDH1A1CYP3A4HPGD
SCHEMBL895951 0.82 MIF (0.64) MIFTRPA1ALDH1A1CYP3A4HPGD
SCHEMBL8763362 0.81 MIF (0.68) MIFTRPA1ALDH1A1CYP3A4HPGD
SCHEMBL18486425 0.77 CA1 (0.39) MIFTRPA1ALDH1A1CYP3A4HPGD
SCHEMBL1457562 0.77 MIF (1.00) MIFTRPA1ALDH1A1CYP3A4HPGD
SCHEMBL14476253 0.77 MIF (0.63) MIFTRPA1ALDH1A1CYP3A4HPGD
SCHEMBL1706732 0.77 MIF (0.63) MIFTRPA1ALDH1A1CYP3A4HPGD
SCHEMBL4780073 0.77 MIF (0.63) MIFTRPA1ALDH1A1CYP3A4HPGD
SCHEMBL10651884 0.77 TRPA1 (0.69) MIFTRPA1ALDH1A1CYP3A4HPGD
SCHEMBL41756 0.77 TRPA1 (1.00) MIFTRPA1ALDH1A1CYP3A4HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1360186-B1 CARBOLINE DERIVATIVES LILLY ICOS LLC (US) 2006-11-22 EP disclosed
US-7122554-B2 Carboline derivatives LILLY ICOS LLC. (US) 2006-10-17 US disclosed
US-20040116458-A1 Chemical compounds LILLY ICOS LLC, A DELAWARE CORPORATION 2004-06-17 US disclosed
EP-1360186-A2 CARBOLINE DERIVATIVES Lilly Icos LLC (US) 2003-11-12 EP disclosed
WO-2002064591-A2 CARBOLINE DERIVATIVES LILLY ICOS LLC (US) 2002-08-22 WO disclosed