SCHEMBL5790701

SCHEMBL5790701

Cc1ccc(C2(C(=O)O)CC=CC2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.47
CYP2C19 P33261 2/20 0.44
AKR1C1 Q04828 1/20 0.42
CYP1A2 P05177 1/20 0.41
HSD11B1 P28845 2/20 0.40
ALDH1A1 P00352 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
OPRM1 P35372 1/20 0.40
LMNA P02545 2/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CCR2 P41597 1/20 0.38
TSHR P16473 1/20 0.38
CES2 O00748 2/20 0.37
CES1 P23141 2/20 0.37
SRD5A2 P31213 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL351393 0.83 AKR1C1 (0.55) CYP2C19AKR1C1CYP1A2HSD11B1ALDH1A1
SCHEMBL16113395 0.81 HDAC4 (0.68) HDAC4CYP2C19AKR1C1HSD11B1ALDH1A1
SCHEMBL3485961 0.80 AKR1C1 (0.62) HDAC4CYP2C19AKR1C1CYP1A2HSD11B1
SCHEMBL1048151 0.80 AKR1C1 (0.68) HDAC4CYP2C19AKR1C1CYP1A2HSD11B1
SCHEMBL15912397 0.78 CYP2C19 (0.50) CYP2C19AKR1C1CYP1A2HSD11B1CYP3A4
SCHEMBL3821416 0.78 AKR1C1 (0.66) HDAC4CYP2C19AKR1C1CYP1A2HSD11B1
SCHEMBL2860893 0.78 AKR1C1 (0.66) HDAC4CYP2C19AKR1C1CYP1A2HSD11B1
SCHEMBL10146430 0.78 LMNA (0.44) CYP2C19AKR1C1CYP1A2HSD11B1ALDH1A1
SCHEMBL16730897 0.77 CYP2C19 (0.43) CYP2C19AKR1C1CYP1A2HSD11B1ALDH1A1
SCHEMBL9685778 0.77 CYP2C19 (0.49) CYP2C19AKR1C1CYP1A2HSD11B1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2968207-A1 HISTONE DEACETYLASE INHIBITORS AND COMPOSITIONS CHDI Foundation, Inc. (US) 2016-01-20 EP disclosed
WO-2014159218-A1 HISTONE DEACETYLASE INHIBITORS AND COMPOSITIONS CHDI FOUNDATION, INC. (US) 2014-10-02 WO disclosed
WO-2006014664-A2 CYCLOPENTYLAMINE AND CYCLOHEXYLAMINE DERIVATIVES AS NK-1/SSRI ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2006-02-09 WO disclosed