SCHEMBL5790992

SCHEMBL5790992

CC(C)(C)CN(NC(=O)c1ccc(CN2CCNCC2)cc1)c1ccnc(C#N)n1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSK P43235 12/20 0.47
CTSL P07711 2/20 0.47
CTSS P25774 2/20 0.47
CTSB P07858 1/20 0.47
GPR4 P46093 2/20 0.40
CHRM3 P20309 1/20 0.40
TBK1 Q9UHD2 2/20 0.39
IKBKE Q14164 1/20 0.39
ABL1 P00519 1/20 0.38
KIT P10721 1/20 0.38
BCR P11274 1/20 0.38
LRRK2 Q5S007 1/20 0.38
F10 P00742 1/20 0.37
ACVR1 Q04771 1/20 0.37
JAK2 O60674 1/20 0.37
JAK3 P52333 1/20 0.37
ITGB3 P05106 1/20 0.37
ITGA2B P08514 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5500170 0.90 CTSK (0.58) CTSKCTSLCTSSCTSBGPR4
SCHEMBL8270732 0.90 CTSK (0.47) CTSKCTSLCTSSCTSBJAK2
SCHEMBL8270035 0.89 CTSK (0.51) CTSKCTSLCTSSCTSBGPR4
SCHEMBL14004314 0.88 ABL1 (0.41) CTSKCTSLCTSSCTSBCHRM3
Trifluoroacetic Acid SCHEMBL3317688 0.86 CTSK (0.54) CTSKCTSLCTSSCTSBGPR4
Trifluoroacetic Acid SCHEMBL5794393 0.85 CTSK (0.44) CTSKCTSLCTSSCTSBACVR1
SCHEMBL8270467 0.84 CTSK (0.48) CTSKCTSLCTSSCTSBGPR4
SCHEMBL5793222 0.81 CTSK (0.41) CTSKCTSLCTSSCTSBGPR4
SCHEMBL5791503 0.80 CTSK (0.47) CTSKCTSLCTSSCTSBGPR4
SCHEMBL8270522 0.80 CTSK (0.51) CTSKCTSLCTSSCTSBGPR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006027211-A1 2,4-SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-03-16 WO claimed
WO-2008112156-A1 CHEMOKINE RECEPTOR MODULATORS ALTIRIS THERAPEUTICS (US) 2008-09-18 WO disclosed
WO-2006027211-A1 2,4-SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-03-16 WO disclosed