SCHEMBL5791503

SCHEMBL5791503

CC(C)(C)CN(NC(=O)c1ccc(F)cc1)c1ccnc(C#N)n1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSK P43235 11/20 0.47
IDO1 P14902 1/20 0.39
CTSL P07711 4/20 0.38
FGFR4 P22455 1/20 0.36
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
CTSB P07858 2/20 0.35
CTSS P25774 2/20 0.35
GPR4 P46093 1/20 0.35
HTT P42858 1/20 0.35
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
CTSC P53634 1/20 0.34
EGLN2 Q96KS0 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8270779 0.90 CTSK (0.40) CTSKIDO1CTSLFGFR4ALDH1A1
SCHEMBL5790636 0.89 CTSK (0.44) CTSKCTSLFGFR4CTSBCTSS
SCHEMBL8271448 0.88 CTSK (0.46) CTSKCTSLFGFR4HTTHDAC1
SCHEMBL8270467 0.88 CTSK (0.48) CTSKCTSLFGFR4HPGDCTSB
SCHEMBL8268844 0.88 CTSK (0.45) CTSKCTSLFGFR4ALDH1A1CTSB
SCHEMBL8271447 0.87 CTSK (0.43) CTSKFGFR4HDAC3HDAC1HDAC2
SCHEMBL8270485 0.86 CTSK (0.37) CTSKIDO1CTSLFGFR4ALDH1A1
SCHEMBL5791384 0.85 CTSK (0.45) CTSKFGFR4CTSSHTT
SCHEMBL8270696 0.85 CTSL (0.47) CTSKIDO1CTSLFGFR4ALDH1A1
SCHEMBL5793878 0.84 CTSK (0.37) CTSKIDO1CTSLCTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006027211-A1 2,4-SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-03-16 WO claimed
WO-2006027211-A1 2,4-SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-03-16 WO disclosed