SCHEMBL5791308

SCHEMBL5791308

O=C(O)CC(=O)OCCc1c[nH]c2ccc(F)cc12

nearest known ligand 0.61

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.61
MPO P05164 12/20 0.57
NOTUM Q6P988 2/20 0.57
MTNR1A P48039 1/20 0.57
MTNR1B P49286 1/20 0.57
SLC6A4 P31645 4/20 0.56
SPR P35270 1/20 0.55
HTR2A P28223 1/20 0.53
TRPM8 Q7Z2W7 1/20 0.53
HTR1A P08908 2/20 0.53
KMT2A Q03164 1/20 0.52
GPR84 Q9NQS5 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5791310 0.94 MPO (0.61) TSHRMPONOTUMMTNR1AMTNR1B
SCHEMBL28364289 0.83 MPO (0.69) TSHRMPONOTUMMTNR1AMTNR1B
SCHEMBL9293385 0.82 MEN1 (0.68) TSHRKMT2A
SCHEMBL4463076 0.80 MPO (0.67) TSHRMPONOTUMMTNR1AMTNR1B
SCHEMBL29902243 0.80 MPO (0.76) TSHRMPONOTUMMTNR1AMTNR1B
SCHEMBL3655654 0.80 MPO (0.76) TSHRMPONOTUMMTNR1AMTNR1B
SCHEMBL351449 0.78 MPO (0.69) TSHRMPONOTUMMTNR1AMTNR1B
SCHEMBL5203631 0.78 MPO (0.80) TSHRMPONOTUMMTNR1AMTNR1B
SCHEMBL2260803 0.77 TSHR (1.00) TSHRMPONOTUMMTNR1AMTNR1B
SCHEMBL20242784 0.76 NOTUM (0.78) TSHRMPONOTUMMTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1651637-A1 3-AMINO CHROMAN AND 2-AMINO TETRALIN DERIVATIVES Wyeth (US) 2006-05-03 EP disclosed
WO-2005012291-A1 3-AMINO CHOMAN AND 2-AMINO TETRALIN DERIVATIVES WYETH (US) 2005-02-10 WO disclosed