Isoniazid

Isoniazid

SCHEMBL5791571

C=C1c2cccc(O)c2C(O)=C2C(=O)[C@]3(O)C(=O)/C(=C(/N)O)C(=O)[C@@H](N(C)C)[C@@H]3[C@@H](O)[C@H]12.NNC(=O)c1ccncc1

nearest known ligand 0.61

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

inhA

The experimentally established mechanism targets of Isoniazid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 12/20 0.61
KDM4E B2RXH2 9/20 0.61
USP2 O75604 9/20 0.61
RECQL P46063 7/20 0.61
HPGD P15428 7/20 0.61
HSD17B10 Q99714 7/20 0.61
THRB P10828 6/20 0.61
LMNA P02545 3/20 0.61
NR1I2 O75469 2/20 0.61
SIRT5 Q9NXA8 2/20 0.61
MC4R P32245 1/20 0.61
L3MBTL1 Q9Y468 7/20 0.61
MEN1 O00255 6/20 0.61
KMT2A Q03164 6/20 0.61
MAPT P10636 5/20 0.61
POLB P06746 3/20 0.61
RAD52 P43351 1/20 0.61
ALDH1A1 P00352 6/20 0.42
HIF1A Q16665 3/20 0.42
TSHR P16473 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL20398184 0.89 TDP1 (0.71) TDP1KDM4EUSP2RECQLHPGD
SCHEMBL4015 0.89 TDP1 (0.73) TDP1KDM4EUSP2RECQLHPGD
Methacycline SCHEMBL5791578 0.79 TDP1 (0.57) TDP1KDM4EUSP2RECQLHPGD
SCHEMBL26628251 0.77 TDP1 (1.00) TDP1KDM4EUSP2RECQLHPGD
SCHEMBL26597994 0.77 TDP1 (1.00) TDP1KDM4EUSP2RECQLHPGD
SCHEMBL30567156 0.77 TDP1 (1.00) TDP1KDM4EUSP2RECQLHPGD
SCHEMBL19555132 0.77 TDP1 (1.00) TDP1KDM4EUSP2RECQLHPGD
SCHEMBL29537520 0.77 TDP1 (1.00) TDP1KDM4EUSP2RECQLHPGD
Hydrochloric Acid SCHEMBL29413670 0.76 TDP1 (1.00) TDP1KDM4EUSP2RECQLHPGD
SCHEMBL12841672 0.76 TDP1 (0.62) TDP1KDM4EUSP2RECQLHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006021833-A2 BISBENZAMIDINES FOR THE TREATMENT OF PNEUMONIA UNIVERSITY OF CINCINNATI (US) 2006-03-02 WO disclosed
US-20040009126-A1 Inhalation system for prevention and treatment of intracellular infections TRANSAVE, INC. (US) 2004-01-15 US disclosed