SCHEMBL5791960

SCHEMBL5791960

Cc1cnc(Cc2ccccc2C(N)=O)cn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.38
CD38 P28907 4/20 0.38
AURKA O14965 1/20 0.38
RPS6KB1 P23443 1/20 0.38
AR P10275 1/20 0.36
CYP2D6 P10635 1/20 0.36
HRH1 P35367 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
MAPT P10636 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36
AKR1C1 Q04828 1/20 0.36
PDE10A Q9Y233 1/20 0.35
HTT P42858 1/20 0.35
NR1I2 O75469 1/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1767524 0.83 TDP1 (0.46) CD38MEN1KMT2AMAPTKDM4E
SCHEMBL28213057 0.78 TSHR (0.42) PARP1AURKARPS6KB1MEN1KMT2A
SCHEMBL15926013 0.76 CYP1A2 (0.43) ARCYP2D6HRH1MEN1KMT2A
SCHEMBL15389131 0.75 NPC1 (0.43) PARP1ARCYP2D6MEN1KMT2A
SCHEMBL29818128 0.75 PARP10 (0.48) PARP1AURKARPS6KB1HRH1KDM4E
SCHEMBL166483 0.75 PARP10 (0.48) PARP1AURKARPS6KB1HRH1KDM4E
SCHEMBL31038176 0.75 JAK2 (0.44) AURKARPS6KB1
SCHEMBL28778421 0.75 JAK2 (0.44) AURKARPS6KB1
SCHEMBL7134588 0.75 TSHR (0.54) PARP1MEN1KMT2AMAPTKDM4E
SCHEMBL13562419 0.73 CYP1A2 (0.46) CYP2D6HRH1KMT2AALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2592070-A2 Tetrazole-substituted arylamides F. Hoffmann-La Roche AG (CH) 2013-05-15 EP disclosed
WO-2006011719-A1 N-SUBSTITUTED-SULFAMOYLBENZOIC ACID DERIVATIVES, METHOD FOR PREPARING THEREOF AND ANTIVIRAL PHARMACEUTICAL COMPOSITION COMPRISING THE SAME B & C BIOPHARM CO., LTD. (KR) 2006-02-02 WO disclosed