SCHEMBL5794080

SCHEMBL5794080

CC(C)CN(NC1CCCCC1)c1ccnc(C#N)n1

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CTSK P43235 14/20 0.51
CTSL P07711 5/20 0.36
CTSB P07858 3/20 0.36
GPR4 P46093 2/20 0.35
CTSS P25774 7/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8270728 0.84 CTSK (0.42) CTSKCTSLCTSBCTSS
SCHEMBL5791767 0.82 CTSK (0.40) CTSKCTSLCTSBGPR4CTSS
SCHEMBL5794349 0.81 CTSK (0.39) CTSKCTSLCTSBGPR4CTSS
SCHEMBL5794370 0.80 CTSK (0.38) CTSKCTSLCTSBGPR4CTSS
SCHEMBL5792335 0.79 CTSK (0.37) CTSKCTSLCTSBCTSS
Trifluoroacetic Acid SCHEMBL5792736 0.78 CTSK (0.38) CTSKCTSLCTSBCTSS
SCHEMBL8270526 0.78 CTSK (0.36) CTSKCTSLCTSBCTSS
SCHEMBL5791458 0.78 KMT2A (0.41) CTSKCTSLCTSBCTSS
SCHEMBL8269410 0.76 CTSK (0.39) CTSKCTSLCTSBGPR4CTSS
SCHEMBL2227354 0.75 CTSK (0.53) CTSKGPR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006027211-A1 2,4-SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-03-16 WO claimed
WO-2006027211-A1 2,4-SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-03-16 WO disclosed