SCHEMBL5794340

SCHEMBL5794340

Cc1nc2ccc(-c3ccc(Cl)cc3Cl)cc2c(=O)n1C[C@H]1CCCN(C(C)C)C1

nearest known ligand 0.82

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 14/20 0.82
CYP2D6 P10635 7/20 0.82
KCNH2 Q12809 10/20 0.67
CYP3A4 P08684 1/20 0.67
HTR2C P28335 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5792960 0.91 CYP2D6 (0.82) GHSRCYP2D6KCNH2CYP3A4HTR2C
SCHEMBL2742703 0.90 GHSR (1.00) GHSRCYP2D6KCNH2CYP3A4HTR2C
SCHEMBL12584175 0.90 GHSR (1.00) GHSRCYP2D6KCNH2CYP3A4HTR2C
SCHEMBL5793061 0.87 CYP2D6 (0.66) GHSRCYP2D6KCNH2CYP3A4HTR2C
SCHEMBL16302710 0.85 GHSR (0.86) GHSRCYP2D6KCNH2CYP3A4
SCHEMBL10077169 0.84 GHSR (0.84) GHSRCYP2D6KCNH2CYP3A4
SCHEMBL5794498 0.84 CYP2D6 (0.82) GHSRCYP2D6KCNH2CYP3A4HTR2C
SCHEMBL5791730 0.81 GHSR (0.73) GHSRCYP2D6KCNH2CYP3A4
SCHEMBL5823257 0.80 GHSR (0.80) GHSRCYP2D6KCNH2CYP3A4HTR2C
SCHEMBL5823255 0.80 GHSR (0.80) GHSRCYP2D6KCNH2CYP3A4HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006012577-A2 QUINAZOLINONE DERIVATIVES USEFUL FOR THE REGULATION OF GLUCOSE HOMEOSTASIS AND FOOD INTAKE BAYER PHARMACEUTICALS CORPORATION (US) 2006-02-02 WO claimed