SCHEMBL5794403

SCHEMBL5794403

CC(O)(CC(N)OCc1cc(Br)cc(Br)c1)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 11/20 0.43
SLC6A4 P31645 2/20 0.36
SLC6A3 Q01959 2/20 0.36
IDO1 P14902 1/20 0.36
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
MAPK1 P28482 1/20 0.34
NR3C2 P08235 1/20 0.33
KMT2A Q03164 2/20 0.33
SLC1A3 P43003 2/20 0.33
SLC1A2 P43004 2/20 0.33
SLC1A1 P43005 2/20 0.33
MEN1 O00255 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
ESR2 Q92731 1/20 0.32
CACNA1F O60840 1/20 0.32
CACNA1D Q01668 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5793923 0.90 IDO1 (0.44) IDO1NR3C2CYP2C19
SCHEMBL5791679 0.88 CHRM3 (0.39) TACR1SLC6A4SLC6A3IDO1KDM4E
SCHEMBL5791672 0.86 TACR1 (0.46) TACR1SLC6A4SLC6A3IDO1KDM4E
SCHEMBL5792856 0.86 SLC1A3 (0.44) TACR1SLC6A4SLC6A3IDO1KDM4E
SCHEMBL5794077 0.85 TACR1 (0.47) TACR1CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL5790217 0.83 TACR1 (0.57) TACR1IDO1CACNA1FCACNA1DCACNA1S
SCHEMBL5790274 0.80 IDO1 (0.45) TACR1IDO1KDM4ELMNAMAPK1
SCHEMBL5793829 0.80 IDO1 (0.42) SLC6A4SLC6A3IDO1KDM4ELMNA
SCHEMBL5793858 0.80 CHRNB2 (0.47) SLC6A4IDO1LMNAMAPK1KMT2A
SCHEMBL5790287 0.80 SLC6A4 (0.44) TACR1SLC6A4SLC6A3IDO1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006014942-A1 ARYLOXYALKYLAMINE NK-1/SSRI INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2006-02-09 WO disclosed