SCHEMBL579506

SCHEMBL579506

NC(=O)c1ccc(Oc2ccc(CCNCc3ccccc3)cc2)cc1.O=C(O)c1ccno1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 15/20 0.76
OPRD1 P41143 13/20 0.76
OPRK1 P41145 10/20 0.76
GRIN2D O15399 1/20 0.62
GRIN3B O60391 1/20 0.62
SLC6A2 P23975 1/20 0.62
SLC6A3 Q01959 1/20 0.62
GRIN1 Q05586 1/20 0.62
KCNH2 Q12809 1/20 0.62
GRIN2A Q12879 1/20 0.62
GRIN2B Q13224 1/20 0.62
ROCK1 Q13464 1/20 0.62
GRIN2C Q14957 1/20 0.62
GRIN3A Q8TCU5 1/20 0.62
LTA4H P09960 1/20 0.50
EPHX2 P34913 1/20 0.50
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
ATM Q13315 1/20 0.48
KDM4E B2RXH2 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL579508 0.90 OPRM1 (0.58) OPRM1OPRD1OPRK1GRIN2DGRIN3B
SCHEMBL580098 0.87 OPRM1 (1.00) OPRM1OPRD1OPRK1GRIN2DGRIN3B
SCHEMBL3692341 0.87 OPRM1 (1.00) OPRM1OPRD1OPRK1GRIN2DGRIN3B
Thiophene Carboxylic Acid SCHEMBL5738716 0.83 OPRM1 (0.57) OPRM1OPRD1OPRK1GRIN2DGRIN3B
SCHEMBL579507 0.81 OPRM1 (0.56) OPRM1OPRD1OPRK1GRIN2DGRIN3B
SCHEMBL3700420 0.79 OPRM1 (0.79) OPRM1OPRD1OPRK1GRIN2DGRIN3B
SCHEMBL3690849 0.78 OPRM1 (0.82) OPRM1OPRD1OPRK1GRIN2DGRIN3B
SCHEMBL5751517 0.78 OPRM1 (0.72) OPRM1OPRD1OPRK1GRIN2DGRIN3B
SCHEMBL3698270 0.77 OPRM1 (1.00) OPRM1OPRD1OPRK1GRIN2DGRIN3B
SCHEMBL13285462 0.77 OPRM1 (0.88) OPRM1OPRD1OPRK1GRIN2DGRIN3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1735268-B1 OPIOID RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2012-02-15 EP disclosed