SCHEMBL5796178

SCHEMBL5796178

O=c1n(Cc2ccc(C(F)C(F)F)cc2)nc2c(-c3ccc(Cl)cc3)c(-c3ccc(Cl)cc3)c(Cl)nn12

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 15/20 0.48
CYP3A4 P08684 4/20 0.35
CYP2C9 P11712 3/20 0.35
CYP2C19 P33261 3/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
LMNA P02545 2/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
HTT P42858 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
HTR2C P28335 1/20 0.32
HTR2B P41595 1/20 0.32
SLC16A3 O15427 1/20 0.31
SLC16A1 P53985 1/20 0.31
MCTS1 Q9ULC4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5795343 0.87 CNR1 (0.47) CNR1CYP3A4CYP2C9CYP2C19MEN1
SCHEMBL13114724 0.83 CNR1 (0.54) CNR1CYP3A4CYP2C19MEN1KMT2A
SCHEMBL3550428 0.82 CNR1 (0.59) CNR1CYP3A4CYP2C9CYP2C19LMNA
SCHEMBL5796174 0.82 CNR1 (0.54) CNR1CYP3A4CYP2C9CYP2C19LMNA
SCHEMBL13114751 0.72 CNR1 (0.49) CNR1CYP3A4CYP2C9CYP2C19LMNA
SCHEMBL4806813 0.72 CNR1 (0.73) CNR1CYP3A4CYP2C9CYP2C19MEN1
SCHEMBL13134239 0.72 CNR1 (0.50) CNR1CYP3A4CYP2C9CYP2C19MEN1
SCHEMBL14180979 0.72 CNR1 (0.62) CNR1CYP3A4CYP2C9CYP2C19MEN1
SCHEMBL13114674 0.72 CNR1 (0.50) CNR1CYP3A4CYP2C9CYP2C19LMNA
SCHEMBL3553773 0.71 NOTUM (0.44) CNR1CYP3A4CYP2C9CYP2C19MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1697371-A1 AZABICYCLIC HETEROCYCLES AS CANNABINOID RECEPTOR MODULATORS Bristol-Myers Squibb Company (US) 2006-09-06 EP disclosed
WO-2005063762-A1 AZABICYCLIC HETEROCYCLES AS CANNABINOID RECEPTOR MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2005-07-14 WO disclosed