SCHEMBL5796837

SCHEMBL5796837

CN(CCCN(C)Cc1cccc2ccccc12)Cc1ccc2ccccc2c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.59
CYP1A2 P05177 2/20 0.59
CYP2C19 P33261 2/20 0.59
SIGMAR1 Q99720 3/20 0.56
LMNA P02545 3/20 0.56
NR1I2 O75469 2/20 0.56
SLC6A2 P23975 2/20 0.56
HTR2A P28223 2/20 0.56
SLC6A4 P31645 2/20 0.56
KCNH2 Q12809 2/20 0.56
ADRA2A P08913 1/20 0.56
ACHE P22303 1/20 0.56
MC5R P33032 5/20 0.50
MC4R P32245 4/20 0.50
MC1R Q01726 4/20 0.50
MC3R P41968 3/20 0.50
MAPK1 P28482 2/20 0.50
PYCR1 P32322 1/20 0.50
KMT2A Q03164 2/20 0.47
DRD2 P14416 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11887346 0.87 CYP2D6 (0.79) CYP2D6CYP1A2CYP2C19SIGMAR1LMNA
SCHEMBL4363764 0.83 BCHE (0.49) CYP2D6CYP1A2CYP2C19SIGMAR1MC5R
SCHEMBL4823146 0.80 CYP2D6 (0.50) CYP2D6CYP1A2CYP2C19SIGMAR1LMNA
SCHEMBL16256972 0.79 CYP2D6 (0.71) CYP2D6CYP1A2CYP2C19SIGMAR1LMNA
SCHEMBL14149518 0.79 SIGMAR1 (0.63) CYP1A2SIGMAR1SLC6A2SLC6A4ACHE
SCHEMBL18085060 0.78 CYP2D6 (0.65) CYP2D6CYP1A2CYP2C19SIGMAR1LMNA
SCHEMBL8088645 0.78 SIGMAR1 (0.61) CYP1A2SIGMAR1SLC6A2SLC6A4ACHE
SCHEMBL10932466 0.77 CYP2D6 (1.00) CYP2D6CYP1A2CYP2C19SIGMAR1LMNA
SCHEMBL6465969 0.76 PYCR1 (0.61) CYP1A2SIGMAR1SLC6A2SLC6A4ACHE
SCHEMBL13381683 0.76 CYP2D6 (0.76) CYP2D6CYP1A2CYP2C19SIGMAR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1644337-A1 MELANOCORTIN-4 RECEPTOR BINDING COMPOUNDS AND METHODS OF USE THEREOF Gene Logic, Inc. (US) 2006-04-12 EP disclosed
WO-2005121100-A1 MELANOCORTIN-4 RECEPTOR BINDING COMPOUNDS AND METHODS OF USE THEREOF GENE LOGIC INC. (US) 2005-12-22 WO disclosed