SCHEMBL5799043

SCHEMBL5799043

Cc1cn2cc(CN)nc2s1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDE8B O95263 1/20 0.43
CYP19A1 P11511 1/20 0.42
TPH1 P17752 16/20 0.39
TPH2 Q8IWU9 16/20 0.39
GHSR Q92847 1/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL2433651 0.76 KDM4E (0.49) PDE8BCYP19A1TPH1TPH2GHSR
SCHEMBL3459088 0.76 CYP19A1 (0.49) PDE8BCYP19A1TPH1TPH2TP53
Bromide SCHEMBL10970945 0.74 CYP19A1 (0.47) PDE8BCYP19A1TPH1TPH2TP53
SCHEMBL12984857 0.73 TPH1 (0.51) CYP19A1TPH1TPH2GHSRMAPT
SCHEMBL12617259 0.68 CYP19A1 (0.43) PDE8BCYP19A1TPH1TPH2
SCHEMBL2386978 0.68 SMN1; SMN2 (0.53) TP53
SCHEMBL17863729 0.67 CYP19A1 (0.45) PDE8BCYP19A1TPH1TPH2GHSR
SCHEMBL23530839 0.66 ALOX15 (0.62) TP53MAPT
SCHEMBL11030523 0.64 TP53 (0.59) CYP19A1TP53MAPT
SCHEMBL23530863 0.64 NPC1 (0.50) TP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006065755-A2 QUATERNARY AMMONIUM SALTS OF FUSED HETEAROMATIC AMINES AS NOVEL MUSCARINIC ACETYLCHOLINE RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2006-06-22 WO disclosed
WO-2003035615-A2 TYROSINE KINASE INHIBITORS MERCK & CO., INC. (US) 2003-05-01 WO disclosed