Oxypurinol

Oxypurinol

SCHEMBL5799552

O.Oc1nc(O)c2cn[nH]c2n1.Oc1nc(O)c2cn[nH]c2n1

nearest known ligand 0.37

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

XDH

The experimentally established mechanism targets of Oxypurinol. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH known ✓ P47989 4/20 0.35
SMN1; SMN2 Q16637 2/20 0.37
RET P07949 1/20 0.35
PI4KA P42356 1/20 0.35
LRRK2 Q5S007 1/20 0.35
PI4K2B Q8TCG2 1/20 0.35
PI4K2A Q9BTU6 1/20 0.35
PI4KB Q9UBF8 1/20 0.35
CDK2 P24941 2/20 0.34
HSP90AA1 P07900 1/20 0.34
IDO1 P14902 1/20 0.34
FGFR1 P11362 1/20 0.34
FGFR2 P21802 1/20 0.34
FGFR3 P22607 1/20 0.34
CYP1A2 P05177 2/20 0.33
ALDH1A1 P00352 2/20 0.33
ADORA2A P29274 2/20 0.33
LMNA P02545 1/20 0.33
TSHR P16473 1/20 0.33
SLC6A4 P31645 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxypurinol SCHEMBL8905877 0.98 SMN1; SMN2 (0.36) SMN1; SMN2XDHRETPI4KALRRK2
Oxypurinol SCHEMBL8905835 0.96 SMN1; SMN2 (0.37) SMN1; SMN2XDHRETPI4KALRRK2
Oxypurinol SCHEMBL8905476 0.96 SMN1; SMN2 (0.37) SMN1; SMN2XDHRETPI4KALRRK2
Oxypurinol SCHEMBL8905886 0.96 SMN1; SMN2 (0.37) SMN1; SMN2XDHRETPI4KALRRK2
Oxypurinol SCHEMBL9421596 0.87 JAK2 (0.40) SMN1; SMN2XDHALDH1A1ADORA2ALMNA
Oxypurinol SCHEMBL9421598 0.87 SMN1; SMN2 (0.36) SMN1; SMN2XDHRETPI4KALRRK2
Oxypurinol SCHEMBL5800677 0.82 SMN1; SMN2 (0.35) SMN1; SMN2CDK2CYP1A2ALDH1A1LMNA
SCHEMBL1952036 0.78 SMN1; SMN2 (0.36) SMN1; SMN2XDHRETPI4KALRRK2
SCHEMBL2266999 0.78 PLK4 (0.45) SMN1; SMN2XDHRETPI4KALRRK2
SCHEMBL8141335 0.78 XDH (0.34) SMN1; SMN2XDHRETPI4KALRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006083687-A1 CRYSTAL SALT OF XANTHINE OXIDASE INHIBITORS CARDIOME PHARMA CORP. (CA) 2006-08-10 WO disclosed