SCHEMBL5799790

SCHEMBL5799790

Cc1cccc2sc(C(N)/C(=C/c3ccc(C(=O)O)cc3)CCOc3cccc4ccccc34)nc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 12/20 0.41
BCL2 P10415 2/20 0.41
BCL2L1 Q07817 2/20 0.41
BAD Q92934 2/20 0.41
PIN1 Q13526 2/20 0.39
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
MAPT P10636 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
CDC7 O00311 1/20 0.35
EEF2K O00418 1/20 0.35
DAPK3 O43293 1/20 0.35
MAP4K4 O95819 1/20 0.35
PAK4 O96013 1/20 0.35
RPS6KB1 P23443 1/20 0.35
MARK3 P27448 1/20 0.35
AXL P30530 1/20 0.35
AKT2 P31751 1/20 0.35
CSNK1A1 P48729 1/20 0.35
MAPKAPK2 P49137 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5823605 0.88 MCL1 (0.41) MCL1BCL2BCL2L1BADPIN1
SCHEMBL5799061 0.83 SCD (0.41) MCL1BCL2BCL2L1BADPIN1
SCHEMBL5808425 0.81 MAPT (0.42) MCL1PIN1KMT2AMEN1MAPT
SCHEMBL5799794 0.79 MCL1 (0.41) MCL1BCL2BCL2L1BADPIN1
SCHEMBL5813649 0.78 MRGPRX4 (0.43) MCL1BCL2BCL2L1BADPIN1
SCHEMBL5797679 0.77 KMT2A (0.41) MCL1BCL2BCL2L1BADPIN1
SCHEMBL5812469 0.77 KMT2A (0.39) MCL1PIN1KMT2AMEN1MAPT
SCHEMBL5810719 0.72 MAPT (0.41) MCL1BCL2BCL2L1BADKMT2A
SCHEMBL5810724 0.72 MAPT (0.41) MCL1BCL2BCL2L1BADKMT2A
SCHEMBL5808413 0.72 PIN1 (0.42) MCL1PIN1KMT2AMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006025683-A1 ARYLAMINOMETHYL PROPENYL BENZHYDROXYAMID DERIVATIVES WITH INHIBITORY ACTIVITY AGAINST HISTONE DEACETYLASE AND METHOD FOR THE PREPARATION THEREOF KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2006-03-09 WO disclosed