SCHEMBL5800531

SCHEMBL5800531

CCc1cc(-n2ccnc2)ccc1C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.52
PDE4B Q07343 2/20 0.52
PDE4C Q08493 2/20 0.52
PDE4D Q08499 2/20 0.52
ADH5 P11766 9/20 0.51
CYP3A4 P08684 1/20 0.50
BAZ2B Q9UIF8 1/20 0.50
DHODH Q02127 1/20 0.48
KDM4E B2RXH2 1/20 0.48
MEN1 O00255 1/20 0.48
MITF O75030 1/20 0.48
ALDH1A1 P00352 1/20 0.48
MAPT P10636 1/20 0.48
KMT2A Q03164 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
TBXAS1 P24557 2/20 0.47
HTT P42858 1/20 0.47
CYP4Z1 Q86W10 1/20 0.46
MAOB P27338 1/20 0.45
ENPP2 Q13822 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3850436 0.82 ADH5 (0.67) PDE4APDE4BPDE4CPDE4DADH5
SCHEMBL26614123 0.79 ADH5 (0.54) ADH5CYP3A4BAZ2BDHODHKDM4E
SCHEMBL15924858 0.79 ADH5 (0.64) ADH5CYP3A4BAZ2BDHODHSMN1; SMN2
SCHEMBL12121100 0.79 CYP2D6 (0.60) PDE4APDE4BPDE4CPDE4DADH5
SCHEMBL12316378 0.79 CYP11B1 (0.52) ADH5CYP3A4BAZ2BDHODHKDM4E
SCHEMBL4674986 0.79 PDE4A (0.46) PDE4APDE4BPDE4CPDE4DADH5
SCHEMBL26614180 0.77 ADH5 (0.54) ADH5CYP3A4BAZ2BDHODHKDM4E
SCHEMBL5806043 0.76 CYP11B1 (0.52) ADH5CYP3A4BAZ2BDHODHKDM4E
SCHEMBL14741230 0.76 ADH5 (0.50) PDE4APDE4BPDE4CPDE4DADH5
Propionic Acid SCHEMBL29217936 0.74 CYP3A4 (0.50) PDE4APDE4BPDE4CPDE4DADH5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006058535-A2 NOVEL N-HETEROCYCLIC PLATINUM AND PALLADIUM CARBENE COMPLEXES, PRODUCTION AND USE THEREOF FOR THE PARTIAL OXIDATION OF HYDROCARBONS Technische Universität Dresden (DE) 2006-06-08 WO disclosed
EP-0496237-B1 N-imidazolyl derivatives of substituted tetrahydrocarbazole and cyclohept[b]indole PHARMACIA SPA (IT) 1996-02-14 EP disclosed
US-5246957-A Thromboxane A2 synthesis for cardiovascular disorders FARMITALIA CARLO ERBA S.R.L. (IT) 1993-09-21 US disclosed
US-5238953-A Thromboxane a2 antagonist FARMITALIA CARLO ERBA S.R.L. (IT) 1993-08-24 US disclosed
EP-0510398-A2 N-Imidazolyl derivatives of substituted indole PHARMACIA S.p.A. (IT) 1992-10-28 EP disclosed
EP-0496237-A2 N-imidazolyl derivatives of substituted tetrahydrocarbazole and cyclohept[b]indole PHARMACIA S.p.A. (IT) 1992-07-29 EP disclosed